Drugs / Zenocutuzumab
last change Jul 2025 re-read 2 minutes ago

Zenocutuzumab

also known as MCLA-128 · Bizengri · Zeno · Zenocutuzumab-zbco

Monoclonal antibody

Developed for
breast carcinoma · castration-resistant prostate carcinoma
Investigated by
Partner Therapeutics, Inc. · Merus B.V.

Trials 3 · a red edge is where a trial was stopped

2015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 2 NCT05588609 Nov 2022 → Jul 2025 castration-resistant prostate carcinoma Partner Therapeutics, Inc. Terminated No outcome recorded
Phase 2 NCT03321981 Jan 2018 → Oct 2022 breast carcinoma Merus B.V. Completed No outcome recorded
Phase 2 NCT02912949 Jan 2015 → Dec 2026 expected Partner Therapeutics, Inc. Active not recruiting No outcome recorded
Also used as a comparator or background therapy in 1 trial
PhaseRegistry idDatesIndicationSponsorStatusOutcome
NCT04100694 Background breast cancer, cancer of unknown primary site, cholangiocarcinoma, colorectal cancer +5 Merus B.V. Approved for marketing No outcome recorded

Evidence & citations 8 cited values

Every value below carries the sentence it was read from. 7 sources stand behind the page.

FieldValueCited text
Known as Zenocutuzumab ClinicalTrials.gov intervention name — accepted as the source's own label NCT03321981
1

NCT02912949

Known as Bizengri ChEMBL registry synonym — accepted as the source's own label CHEMBL4298025
Known as MCLA-128 ClinicalTrials.gov intervention name — accepted as the source's own label NCT05588609
1

NCT04100694

Known as Zeno Zenocutuzumab, or Zeno, is a treatment that is being tested to see if it can stop cancer that is growing because of NRG1 gene fusions.” PMID 38348690 Feb 2024
Known as Zenocutuzumab-zbco ChEMBL registry synonym — accepted as the source's own label CHEMBL4298025
Action Inhibit inhibits NRG1 binding” PMID 38348690 Feb 2024
Modality Monoclonal antibody “HER2/HER3 bispecific antibody” NCT04100694
Route Intravenous “750 mg intravenously every 2 weeks” PMID 39908431 Feb 2025