Drugs / Etrolizumab
last change Oct 2023 re-read 2 minutes ago

Etrolizumab

Monoclonal antibody targets ITGB7

Developed for
ulcerative colitis · Crohn disease
Investigated by
Hoffmann-La Roche · Genentech, Inc.

Trials 14 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 14 trials
Phase 1 NCT03478956 Mar 2018 → Dec 2019 Crohn disease, ulcerative colitis Hoffmann-La Roche Terminated No outcome recorded
Phase 1 NCT02996019 Dec 2016 → Apr 2018 Genentech, Inc. Completed No outcome recorded
Phase 1 NCT02629744 Dec 2015 → Jun 2016 Genentech, Inc. Completed No outcome recorded
Phase 1 NCT00694980 Sep 2008 → Sep 2011 ulcerative colitis Genentech, Inc. Completed No outcome recorded
Phase 22 trials
Phase 2 NCT01461317 Nov 2011 → Aug 2016 ulcerative colitis Genentech, Inc. Completed No outcome recorded
Phase 2 NCT01336465 Sep 2011 → Sep 2012 ulcerative colitis Genentech, Inc. Completed No outcome recorded
Phase 38 trials
Phase 3 NCT02403323 Jun 2015 → Oct 2023 Crohn disease Hoffmann-La Roche Terminated No outcome recorded
Phase 3 NCT02394028 Mar 2015 → Sep 2021 Crohn disease Hoffmann-La Roche Completed No outcome recorded
Phase 3 NCT02136069 Dec 2014 → Jun 2020 ulcerative colitis Hoffmann-La Roche Completed No outcome recorded
Phase 3 NCT02171429 Nov 2014 → Mar 2020 ulcerative colitis Hoffmann-La Roche Completed No outcome recorded
Phase 3 NCT02163759 Nov 2014 → Feb 2020 ulcerative colitis Hoffmann-La Roche Completed No outcome recorded
Phase 3 NCT02118584 Sep 2014 → Oct 2023 ulcerative colitis Hoffmann-La Roche Terminated No outcome recorded
Phase 3 NCT02165215 Aug 2014 → Apr 2020 ulcerative colitis Hoffmann-La Roche Completed No outcome recorded
Phase 3 NCT02100696 May 2014 → Apr 2020 ulcerative colitis Hoffmann-La Roche Completed No outcome recorded

Press releases naming this drug 1 release

DateIssuerRelease
2020-08-10 Roche Global Development Roche provides update on phase III studies of etrolizumab in people with moderately to severely active ulcerative colitis roche.com

Evidence & citations 11 cited values

Every value below carries the sentence it was read from. 16 sources stand behind the page.

FieldValueCited text
Known as Etrolizumab “BACKGROUND: Etrolizumab is a humanised monoclonal antibody that selectively binds the β7 subunit of the heterodimeric integrins α4β7 and αEβ7.” PMID 24814090 May 2014
12

Etrolizumab is a gut-targeted, anti-β7 integrin, monoclonal antibody.” PMID 34798039 Nov 2021

NCT02403323

NCT02136069

NCT01461317

NCT02163759

NCT03478956

NCT02118584

NCT02629744

NCT02394028

NCT02171429

NCT02165215

NCT02996019

Known as Anti-.beta.7 ChEMBL registry synonym — accepted as the source's own label CHEMBL1743015
Known as Anti-Beta7 Pro145223 ChEMBL registry synonym — accepted as the source's own label CHEMBL1743015
Known as PRO-145223 ChEMBL registry synonym — accepted as the source's own label CHEMBL1743015
Known as RG-7413 ChEMBL registry synonym — accepted as the source's own label CHEMBL1743015
Known as rhuMAb Beta7 ClinicalTrials.gov intervention name — accepted as the source's own label NCT00694980
Action Inhibit “anti-β7 integrin” PMID 34798039 Nov 2021
Modality Monoclonal antibody “Etrolizumab is a humanised monoclonal antibodyPMID 24814090 May 2014
Route Intravenous Intravenous and subcutaneous escalating doses” NCT00694980
Route Subcutaneous “Intravenous and subcutaneous escalating doses” NCT00694980
Target ITGB7 “Etrolizumab is a novel, dual-action anti-β7 integrin antibody” PMID 33778929 Mar 2021