Drugs / AZD4877
last change Dec 2009 re-read 3 minutes ago

AZD4877

Small molecule targets KIF11 via inhibition

Developed for
acute myeloid leukemia · bladder transitional cell carcinoma · carcinoma · lymphoma · neoplasm · non-Hodgkin lymphoma · renal pelvis carcinoma · ureter cancer
+1 more · urethra cancer
Investigated by
AstraZeneca

Trials 6

200720082009201020112012201320142015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 15 trials · 1 missed
Phase 1 NCT00613652 Jan 2008 → Jun 2009 carcinoma AstraZeneca Completed No outcome recorded
Phase 1 NCT00486265 Jul 2007 → Jul 2009 acute myeloid leukemia AstraZeneca Terminated Missed primary
Phase 1 NCT00471367 Apr 2007 → Dec 2008 non-Hodgkin lymphoma AstraZeneca Terminated No outcome recorded Stop: Enrollment
Phase 1 NCT00460460 Mar → Aug 2007 lymphoma AstraZeneca Terminated No outcome recorded Stop: Enrollment
Phase 1 NCT00389389 Sep 2006 → Aug 2008 neoplasm AstraZeneca Completed No outcome recorded
Phase 21 trial · 1 missed
Phase 2 NCT00661609 May 2008 → May 2009 bladder transitional cell carcinoma, renal pelvis carcinoma, ureter cancer, urethra cancer AstraZeneca Completed Missed primary

Evidence & citations 5 cited values

Every value below carries the sentence it was read from. 7 sources stand behind the page.

FieldValueCited text
Known as AZD4877 ClinicalTrials.gov intervention name — accepted as the source's own label NCT00460460 ↗
5

NCT00389389 ↗

NCT00613652 ↗

NCT00661609 ↗

NCT00486265 ↗

NCT00471367 ↗

Action Inhibit “AZD4877 is an Eg5 or Kinesin Spindle Protein inhibitor” NCT00471367 ↗
1

“Kinesin-like protein 1 inhibitor” CHEMBL1829433 ↗

Modality Small molecule — CHEMBL1829433 ↗
Route Intravenous “intravenous infusion” NCT00389389 ↗
Target KIF11 “Kinesin-like protein 1 inhibitor” CHEMBL1829433 ↗