Drugs / PF-4191834
last change Feb 2011 re-read 2 minutes ago

PF-4191834

also known as PF-04191834

Small molecule targets ALOX5 via inhibition

Developed for
asthma · osteoarthritis, knee
Investigated by
Pfizer

Trials 2 · a red edge is where a trial was stopped

20082009201020112012201320142015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 2 NCT01147458 Jul 2010 → Feb 2011 osteoarthritis, knee Pfizer Terminated No outcome recorded
Phase 2 NCT00723021 Jul → Dec 2008 asthma Pfizer Completed No outcome recorded
Also used as a comparator or background therapy in 1 trial
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1 NCT01265732 Comparator Dec 2010 → Jan 2011 Pfizer Withdrawn No outcome recorded

Evidence & citations 6 cited values

Every value below carries the sentence it was read from. 4 sources stand behind the page.

FieldValueCited text
Known as PF-4191834 ChEMBL registry synonym — accepted as the source's own label CHEMBL4297416
Known as PF-04191834 ClinicalTrials.gov intervention name — accepted as the source's own label NCT01265732
2

NCT00723021

NCT01147458

Action Inhibit “PF-04191834 works in animal models by inhibiting one of the enzymes, 5-lipoxygenase” NCT01147458
1

“Arachidonate 5-lipoxygenase inhibitor” CHEMBL4297416

Modality Small molecule CHEMBL4297416
Route Oral oral dispersion” NCT00723021
Target ALOX5 “Arachidonate 5-lipoxygenase inhibitor” CHEMBL4297416