Drugs / TEDATIOXETINE
TEDATIOXETINE
also known as
LU AA 24530 HYDROBROMIDE · Lu AA24530 · Lu AA24530 (HBr) · Tedatioxetina · TEDATIOXETINE HYDROBROMIDE
Small molecule targets ADRA1A, HTR2A, HTR2C, SLC6A2, SLC6A3, SLC6A4 via inhibition
Trials 1 · a red edge is where a trial was stopped
| Phase | Registry id | Dates | Indication | Sponsor | Status | Outcome |
|---|---|---|---|---|---|---|
| Phase 2 | NCT00599911 | Oct 2007 → Mar 2009 | major depressive disorder | H. Lundbeck A/S | Completed | No outcome recorded |
Evidence & citations 15 cited values
Every value below carries the sentence it was read from. 2 sources stand behind the page.
| Field | Value | Cited text |
|---|---|---|
| Known as | TEDATIOXETINE | ChEMBL registry synonym — accepted as the source's own label CHEMBL2104986 ↗ |
| Known as | LU AA 24530 HYDROBROMIDE | ChEMBL registry synonym — accepted as the source's own label CHEMBL2104986 ↗ |
| Known as | Lu AA24530 | ClinicalTrials.gov intervention name — accepted as the source's own label NCT00599911 ↗ |
| Known as | Lu AA24530 (HBr) | ChEMBL registry synonym — accepted as the source's own label CHEMBL2104986 ↗ |
| Known as | Tedatioxetina | ChEMBL registry synonym — accepted as the source's own label CHEMBL2104986 ↗ |
| Known as | TEDATIOXETINE HYDROBROMIDE | ChEMBL registry synonym — accepted as the source's own label CHEMBL2104986 ↗ |
| Action | Inhibit | “Serotonin 2a (5-HT2a) receptor antagonist” CHEMBL2104986 ↗5“Serotonin 2c (5-HT2c) receptor antagonist” CHEMBL2104986 ↗ “Alpha-1a adrenergic receptor antagonist” CHEMBL2104986 ↗ “Norepinephrine transporter inhibitor” CHEMBL2104986 ↗ “Serotonin transporter inhibitor” CHEMBL2104986 ↗ “Dopamine transporter inhibitor” CHEMBL2104986 ↗ |
| Modality | Small molecule | — CHEMBL2104986 ↗ |
| Route | Oral | “per oral, once daily for 6 weeks” NCT00599911 ↗ |
| Target | ADRA1A | “Alpha-1a adrenergic receptor antagonist” CHEMBL2104986 ↗ |
| Target | HTR2A | “Serotonin 2a (5-HT2a) receptor antagonist” CHEMBL2104986 ↗ |
| Target | HTR2C | “Serotonin 2c (5-HT2c) receptor antagonist” CHEMBL2104986 ↗ |
| Target | SLC6A2 | “Norepinephrine transporter inhibitor” CHEMBL2104986 ↗ |
| Target | SLC6A3 | “Dopamine transporter inhibitor” CHEMBL2104986 ↗ |
| Target | SLC6A4 | “Serotonin transporter inhibitor” CHEMBL2104986 ↗ |