Drugs / Alcaftadine
last change Mar 2022 re-read 2 minutes ago

Alcaftadine

also known as R89674 · Lastacaft · Alcaftadina

Small molecule targets HRH1 via inhibition

Developed for
conjunctivitis · allergic rhinitis · atopic conjunctivitis
Investigated by
Vistakon Pharmaceuticals · Starx Research Center, LLC

Regulatory milestones approvals, filings & regulatory actions · 2 recorded

MilestoneJurisdictionBrandIndicationDateSentence it was read from
Label expansion US (FDA) LASTACAFT 2021-12-10 fda.gov
Approved US (FDA) LASTACAFT 2010-07-28 fda.gov

Trials 6 · a red edge is where a trial was stopped

2006200720082009201020112012201320142015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 35 trials
Phase 3 NCT00889330 Apr → May 2009 conjunctivitis Vistakon Pharmaceuticals Completed No outcome recorded
Phase 3 NCT00364091 Aug → Oct 2006 conjunctivitis Vistakon Pharmaceuticals Completed No outcome recorded
Phase 3 NCT00241319 Oct → Dec 2005 conjunctivitis Vistakon Pharmaceuticals Completed No outcome recorded
Phase 3 NCT00244543 Oct → Nov 2005 conjunctivitis Vistakon Pharmaceuticals Completed No outcome recorded
Phase 3 NCT00223951 Sep → Dec 2005 Vistakon Pharmaceuticals Completed No outcome recorded
Phase 41 trial
Phase 4 NCT01808768 Apr → Oct 2013 allergic rhinitis, conjunctivitis Starx Research Center, LLC Unknown No outcome recorded
Also used as a comparator or background therapy in 3 trials
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 4 NCT02308501 Comparator Dec 2014 → Feb 2015 conjunctivitis ORA, Inc. Completed No outcome recorded
Phase 4 NCT01732757 Comparator Nov → Dec 2012 atopic conjunctivitis Allergan Completed No outcome recorded
Phase 4 NCT01470118 Comparator Oct → Dec 2011 atopic conjunctivitis Allergan Completed No outcome recorded

Press releases naming this drug 1 release

DateIssuerRelease
2022-03-15 AbbVie Now Available Over the Counter, LASTACAFT® Provides Eye Allergy Itch Relief in Minutes that Lasts Through 16 Hours abbvie.com

Evidence & citations 7 cited values

Every value below carries the sentence it was read from. 10 sources stand behind the page.

FieldValueCited text
Known as alcaftadine ClinicalTrials.gov intervention name — accepted as the source's own label NCT00889330
3

NCT01732757

NCT01808768

NCT01470118

Known as Alcaftadina ChEMBL registry synonym — accepted as the source's own label CHEMBL1201747
Known as Lastacaft “Alcaftadine(Lastacaft™)” NCT01808768
1

NCT02308501

Known as R89674 ClinicalTrials.gov intervention name — accepted as the source's own label NCT00364091
3

NCT00244543

NCT00223951

NCT00241319

Action Inhibit “Histamine H1 receptor antagonist” CHEMBL1201747
Modality Small molecule CHEMBL1201747
Target HRH1 “Histamine H1 receptor antagonist” CHEMBL1201747