Drugs / Theliatinib
last change Dec 2018 re-read 3 minutes ago

Theliatinib

also known as HMPL-309 · Xiliertinib

Small molecule targets EGFR via inhibition

Developed for
cancer
Investigated by
Hutchison Medipharma Limited

Trials 2

201320142015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1 NCT02601274 Apr 2015 → Dec 2018 cancer Hutchison Medipharma Limited Terminated No outcome recorded
Phase 1 NCT02601248 Oct 2012 → Feb 2016 cancer Hutchison Medipharma Limited Completed No outcome recorded

Press releases naming this drug 1 release

DateIssuerRelease
2012-11-01 Hutchison Medipharma Limited Hutchison MediPharma Limited initiates Phase I clinical study with its novel EGFR inhibitor Theliatinib hutch-med.com ↗

Evidence & citations 7 cited values

Every value below carries the sentence it was read from. 3 sources stand behind the page.

FieldValueCited text
Known as Theliatinib ClinicalTrials.gov intervention name — accepted as the source's own label NCT02601274 ↗
1

NCT02601248 ↗

Known as HMPL-309 ChEMBL registry synonym — accepted as the source's own label CHEMBL5314410 ↗
Known as Xiliertinib ChEMBL registry synonym — accepted as the source's own label CHEMBL5314410 ↗
Action Inhibit “EGFR tyrosine kinase inhibitor” NCT02601248 ↗
Modality Small molecule — CHEMBL5314410 ↗
Route Oral “oral,once daily” NCT02601248 ↗
Target EGFR “EGFR tyrosine kinase inhibitor” NCT02601248 ↗