Drugs / Citarinostat
last change Jun 2024 re-read 2 minutes ago

Citarinostat

also known as ACY-241 · CC-96241 · HDAC-IN-2

Small molecule targets HDAC6 via inhibition

Developed for
cancer · melanoma · non-small cell lung carcinoma · plasma cell myeloma · smoldering plasma cell myeloma
Investigated by
Celgene Corporation · ApoCell, Inc. · Celerion · Massachusetts General Hospital · NYU Langone Health · OncoPep, Inc.
+1 more · Syneos Health

Trials 5 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1 NCT02886065 Mar 2017 → Sep 2026 expected smoldering plasma cell myeloma Massachusetts General Hospital Active not recruiting No outcome recorded
Phase 1 NCT02935790 Sep 2016 → Apr 2017 melanoma Celgene Corporation Completed No outcome recorded
Phase 1 NCT02635061 Aug 2016 → Jan 2024 non-small cell lung carcinoma Celgene Corporation Terminated No outcome recorded
Phase 1 NCT02551185 Dec 2015 → Sep 2019 cancer Celgene Corporation Completed No outcome recorded
Phase 1 NCT02400242 May 2015 → Jun 2024 plasma cell myeloma Celgene Corporation Terminated No outcome recorded

Evidence & citations 8 cited values

Every value below carries the sentence it was read from. 7 sources stand behind the page.

FieldValueCited text
Known as Citarinostat “Selective Histone Deacetylase Inhibitor ACY-241 (Citarinostat) Plus Nivolumab in Advanced Non-Small Cell Lung Cancer: Results From a Phase Ib Study.” PMID 34552864 Sep 2021
2

Citarinostat (CC-96241; previously ACY-241), an oral inhibitor of histone deacetylases (HDACs) with selectivity for HDAC6” PMID 35070991 Jan 2022

NCT02886065

Known as ACY-241 “Citarinostat (CC-96241; previously ACY-241), an oral inhibitor of histone deacetylases (HDACs) with selectivity for HDAC6” PMID 35070991 Jan 2022
3

NCT02635061

NCT02935790

NCT02400242

Known as CC-96241 “Citarinostat (CC-96241; previously ACY-241), an oral inhibitor of histone deacetylases (HDACs) with selectivity for HDAC6” PMID 35070991 Jan 2022
Known as HDAC-IN-2 ChEMBL registry synonym — accepted as the source's own label CHEMBL3693786
Action Inhibit “Histone deacetylase inhibitor” NCT02400242
Modality Small molecule “Citarinostat is an orally active, small-molecule Histone Deacetylase (HDAC) Inhibitor” NCT02886065
1

CHEMBL3693786

Route Oral oral ACY-241” NCT02400242
Target HDAC6 “with selectivity for HDAC6PMID 35070991 Jan 2022