Drugs / PEGDINETANIB
last change Jan 2015 re-read 2 minutes ago

PEGDINETANIB

Protein / enzyme biologic targets KDR via inhibition

Developed for
glioblastoma · cancer · neoplasm · colorectal cancer · non-small cell lung carcinoma
Investigated by
Adnexus, A Bristol-Myers Squibb R&D Company · Bristol-Myers Squibb

Trials 4 · a red edge is where a trial was stopped

200720082009201020112012201320142015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 13 trials
Phase 1 NCT01146171 Nov 2013 → Jan 2015 neoplasm Bristol-Myers Squibb Withdrawn No outcome recorded
Phase 1 NCT00768911 Oct 2008 → Oct 2010 glioblastoma Adnexus, A Bristol-Myers Squibb R&D Company Unknown No outcome recorded
Phase 1 NCT00374179 Aug 2006 → Nov 2008 cancer Adnexus, A Bristol-Myers Squibb R&D Company Completed No outcome recorded
Phase 21 trial
Phase 2 NCT00562419 Oct 2007 → Jun 2011 glioblastoma Adnexus, A Bristol-Myers Squibb R&D Company Unknown No outcome recorded
Also used as a comparator or background therapy in 2 trials
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 2 NCT00851045 Comparator Oct 2009 → Sep 2011 colorectal cancer Bristol-Myers Squibb Completed No outcome recorded
Phase 2 NCT00850577 Comparator Jun 2009 → Aug 2013 non-small cell lung carcinoma Bristol-Myers Squibb Terminated No outcome recorded

Evidence & citations 9 cited values

Every value below carries the sentence it was read from. 8 sources stand behind the page.

FieldValueCited text
Known as PEGDINETANIB ChEMBL registry synonym — accepted as the source's own label CHEMBL2108356
Known as Angiocept ChEMBL registry synonym — accepted as the source's own label CHEMBL2108356
Known as BMS-844203 “Phase I and pharmacokinetic study of CT-322 (BMS-844203), a targeted Adnectin inhibitor of VEGFR-2 based on a domain of human fibronectin.” PMID 21224368 Jan 2011
1

NCT01146171

Known as CT-322 “BMS-844203 (CT-322)” NCT01146171
5

NCT00850577

NCT00562419

NCT00768911

NCT00851045

NCT00374179

Known as VEGFR-2 INHIBITOR PEPTIDE CT-322 ChEMBL registry synonym — accepted as the source's own label CHEMBL2108356
Action Inhibit “Vascular endothelial growth factor receptor 2 inhibitor” CHEMBL2108356
1

“a VEGFR-2 inhibitor” PMID 21224368 Jan 2011

Modality Protein / enzyme biologic “the first human fibronectin domain-based targeted biologic (Adnectin) to enter clinical studies” PMID 21224368 Jan 2011
Route Intravenous “Patients with advanced solid malignancies were treated with escalating doses of CT-322 intravenously (i.v.) weekly (qw), or biweekly (q2w).” PMID 21224368 Jan 2011
Target KDR “Vascular endothelial growth factor receptor 2 inhibitor” CHEMBL2108356