Drugs / Fepixnebart
last change Apr 2025 re-read 2 minutes ago

Fepixnebart

also known as LY3016859

Monoclonal antibody targets EREG, TGFA via inhibition

Developed for
chronic pain syndrome · diabetic polyneuropathy · diabetic kidney disease · osteoarthritis · osteoarthritis, knee
Investigated by
Eli Lilly and Company

Trials 6 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 11 trial
Phase 1 NCT01545583 Apr → Sep 2012 Eli Lilly and Company Completed No outcome recorded
Phase 1/21 trial
Phase 1/2 NCT01774981 Mar 2013 → Aug 2015 diabetic kidney disease Eli Lilly and Company Completed No outcome recorded
Phase 24 trials
Phase 2 NCT04529096 Aug 2020 → Jun 2021 chronic pain syndrome Eli Lilly and Company Completed No outcome recorded
Phase 2 NCT04476108 Jul 2020 → Jul 2021 diabetic polyneuropathy Eli Lilly and Company Completed No outcome recorded
Phase 2 NCT04456686 Jul 2020 → Apr 2021 osteoarthritis Eli Lilly and Company Completed No outcome recorded
Phase 2 NCT05986292 Jan 2020 → Apr 2027 expected chronic pain syndrome, diabetic polyneuropathy, osteoarthritis, knee Eli Lilly and Company Recruiting No outcome recorded

Evidence & citations 7 cited values

Every value below carries the sentence it was read from. 6 sources stand behind the page.

FieldValueCited text
Known as Fepixnebart Fepixnebart (LY3016859), a humanized immunoglobulin G4 monoclonal antibody with high binding affinity to epiregulin and tumor growth factor-α, is being developed as a novel...” PMID 40266472 Apr 2025
1

Fepixnebart (LY3016859), a humanized immunoglobulin G4 monoclonal antibody with high binding affinity to epiregulin and tumor growth factor-α, is being developed as a novel...” PMID 40266472 Apr 2025

Known as LY3016859 “Fepixnebart (LY3016859), a humanized immunoglobulin G4 monoclonal antibody with high binding affinity to epiregulin and tumor growth factor-α, is being developed as a novel...” PMID 40266472 Apr 2025
4

NCT01774981

NCT01545583

NCT05986292

NCT04529096

Action Inhibit “Protransforming growth factor alpha inhibitor” CHEMBL4594573
1

“Proepiregulin inhibitor” CHEMBL4594573

Modality Monoclonal antibody “a humanized immunoglobulin G4 monoclonal antibodyPMID 40266472 Apr 2025
1

CHEMBL4594573

Route Intravenous “Administered intravenously” NCT01545583
Target EREG “Proepiregulin inhibitor” CHEMBL4594573
Target TGFA “Protransforming growth factor alpha inhibitor” CHEMBL4594573