Drugs / GAMCEMETINIB
last change May 2026 re-read 2 minutes ago

GAMCEMETINIB

also known as CC-99677 · BMS-986371

Small molecule

Developed for
ankylosing spondylitis
Investigated by
Celgene Corporation · Bristol-Myers Squibb

Trials 7 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 16 trials
Phase 1 NCT05445440 Sep → Nov 2022 Bristol-Myers Squibb Completed No outcome recorded
Phase 1 NCT05284890 May → Jul 2022 Bristol-Myers Squibb Completed No outcome recorded
Phase 1 NCT04958291 Aug → Dec 2021 Celgene Corporation Completed No outcome recorded
Phase 1 NCT04718636 Sep 2020 → Aug 2021 Celgene Corporation Completed No outcome recorded
Phase 1 NCT04268394 Mar 2020 → Jun 2021 Celgene Corporation Completed No outcome recorded
Phase 1 NCT03554993 May 2018 → Jul 2019 Celgene Corporation Completed No outcome recorded
Phase 21 trial
Phase 2 NCT04947579 Aug 2021 → Feb 2023 ankylosing spondylitis Celgene Corporation Terminated No outcome recorded

Evidence & citations 6 cited values

Every value below carries the sentence it was read from. 11 sources stand behind the page.

FieldValueCited text
Known as GAMCEMETINIB ChEMBL registry synonym — accepted as the source's own label CHEMBL5314585
Known as BMS-986371 “CC-99677 (BMS-986371) is a novel, small-molecule covalent inhibitor of mitogen-activated protein kinase-activated protein kinase 2 (MK2).” PMID 42167889 May 2026
1

NCT05445440

Known as CC-99677 ClinicalTrials.gov intervention name — accepted as the source's own label NCT05284890
5

NCT03554993

NCT04718636

NCT04947579

NCT04958291

NCT04268394

Action Inhibit “CC-99677 inhibition of MK2 is a promising approach for the treatment of inflammatory diseases” PMID 35982464 Aug 2022
Modality Small molecule “CC-99677 (BMS-986371) is a novel, small-molecule covalent inhibitor of mitogen-activated protein kinase-activated protein kinase 2 (MK2).” PMID 42167889 May 2026
Route Oral “Dosed orally, CC-99677 is efficacious in a rat model of ankylosing spondylitis.” PMID 35691544 Jun 2022