Drugs / AMXT 1501

Trials 5 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 01 trial
Phase 0 NCT05717153 Oct 2023 → Jan 2027 expected malignant glioma Mayo Clinic Recruiting No outcome recorded
Phase 11 trial
Phase 1 NCT03536728 Jun 2018 → Dec 2022 carcinoma Aminex Therapeutics, Inc. Completed No outcome recorded
Phase 1/23 trials
Phase 1/2 NCT06465199 May 2026 → May 2033 expected Ewing sarcoma, atypical teratoid rhabdoid tumor, diffuse intrinsic pontine glioma, embryonal tumor with multilayered rosettes +2 Milton S. Hershey Medical Center Recruiting No outcome recorded
Phase 1/2 NCT07287917 Jan 2026 → Feb 2028 expected cutaneous melanoma, hormone receptor-positive breast cancer Aminex Therapeutics, Inc. Recruiting No outcome recorded
Phase 1/2 NCT05500508 Nov 2022 → Dec 2024 breast cancer, cervical cancer, colorectal cancer, diffuse midline glioma, H3 K27M-mutant +10 Aminex Therapeutics, Inc. Terminated No outcome recorded
Also used as a comparator or background therapy in 1 trial
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1 NCT03077477 Comparator Jun 2018 neoplasm, poisoning Aminex Therapeutics, Inc. Withdrawn No outcome recorded

Evidence & citations 5 cited values

Every value below carries the sentence it was read from. 8 sources stand behind the page.

FieldValueCited text
Known as AMXT 1501 AMXT 1501 is a polyamine transport inhibitor which prevents uptake of polyamines from the extracellular environment.” NCT05717153
7

“oral AMXT 1501 dicaprate (AMXT1501) in combination with DFMO” NCT03536728

NCT05500508

NCT03077477

NCT05717153

NCT07287917

NCT03536728

NCT06465199

Known as AMXT 1501 dicaprate “The objective of this study is to determine the safety and tolerability of oral AMXT 1501 dicaprate (AMXT1501) in combination with IV DFMO in patients with advanced solid...” NCT05500508
1

“oral AMXT 1501 dicaprate (AMXT1501) in combination with DFMO” NCT03536728

Action Inhibit “AMXT 1501, a potent inhibitor of polyamine transport” PMID 40913836 Sep 2025
Modality Small molecule CHEMBL474635
Route Oral orally administered” NCT03077477