Drugs / Delpazolid
last change Jun 2026 re-read 2 minutes ago

Delpazolid

also known as LCB01-0371 · DZD

Small molecule

Developed for
pulmonary tuberculosis · pulmonary non-tuberculous mycobacterial infection · rifampicin-resistant tuberculosis · staphylococcal infection
Investigated by
LigaChem Biosciences, Inc. · Radboud University Medical Center · University of California, San Francisco · GlaxoSmithKline · Ludwig-Maximilians - University of Munich · University College, London
+32 more · Critical Path Institute · Desmond Tutu TB Centre · European Lung Foundation · European Respiratory Society · Find · German Center for Infection Research · Helmholtz Zentrum München · Instituto de Saude Publica da Universidade do Porto · Janssen, LP · KNCV Tuberculosis Foundation · Korea University · London School of Hygiene and Tropical Medicine · Lygature · Michael Hoelscher · National Institute of Health, Korea · Otsuka Pharmaceutical Development & Commercialization, Inc. · Perinatal HIV Research Unit of the University of the Witswatersrand · Research Center Borstel · Research Institute for Development · Seoul National University · Seoul National University Hospital · TASK Applied Science · TB Alliance · Tuberculosis Network European Trialsgroup · University of Cambridge · University of Hamburg-Eppendorf · University of Liverpool · University of Milano · University of Oxford · University of St Andrews · Uppsala University · Vita-Salute San Raffaele University

Trials 14 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 17 trials
Phase 1 NCT03492996 Jun → Aug 2020 LigaChem Biosciences, Inc. Completed No outcome recorded
Phase 1 NCT02882789 Sep 2016 → Jul 2017 LigaChem Biosciences, Inc. Completed No outcome recorded
Phase 1 NCT02538003 Sep → Dec 2015 LigaChem Biosciences, Inc. Completed No outcome recorded
Phase 1 NCT02529241 Jul → Dec 2015 LigaChem Biosciences, Inc. Terminated No outcome recorded
Phase 1 NCT02540460 Jun → Dec 2014 LigaChem Biosciences, Inc. Completed No outcome recorded
Phase 1 NCT01842516 Mar → Jul 2013 LigaChem Biosciences, Inc. Completed No outcome recorded
Phase 1 NCT01554995 Mar → Dec 2012 LigaChem Biosciences, Inc. Completed No outcome recorded
Phase 26 trials
Phase 2 NCT06004037 Jan 2024 → Sep 2025 pulmonary non-tuberculous mycobacterial infection LigaChem Biosciences, Inc. Completed No outcome recorded
Phase 2 NCT06114628 Jan 2024 → Feb 2027 expected pulmonary tuberculosis University College, London Recruiting No outcome recorded
Phase 2 NCT05807399 Apr 2023 → Oct 2027 expected pulmonary tuberculosis Michael Hoelscher Recruiting No outcome recorded
Phase 2 NCT05225558 Apr 2022 → Feb 2024 staphylococcal infection LigaChem Biosciences, Inc. Terminated No outcome recorded
Phase 2 NCT04550832 Oct 2021 → Jan 2023 pulmonary tuberculosis LigaChem Biosciences, Inc. Completed No outcome recorded
Phase 2 NCT02836483 Dec 2016 → Jul 2019 pulmonary tuberculosis LigaChem Biosciences, Inc. Completed No outcome recorded
Phase 31 trial
Phase 3 NCT07675954 Oct 2026 → Jun 2032 expected rifampicin-resistant tuberculosis Seoul National University Hospital Not yet recruiting No outcome recorded

Evidence & citations 5 cited values

Every value below carries the sentence it was read from. 16 sources stand behind the page.

FieldValueCited text
Known as Delpazolid Delpazolid (LCB01-0371) is a novel oxazolidinone derivative with a good safety profile for treating gram-positive pathogenic infections such as Mycobacterium abscessus, a...” PMID 38436463 Mar 2024
6

“The investigational MDR-END Plus regimen consists of oral anti-tuberculosis drugs including bedaquiline, delamanid, delpazolid, levofloxacin, and pyrazinamide.” NCT07675954

NCT06114628

NCT05807399

NCT04550832

NCT06004037

NCT05225558

Known as DZD “Drug: Delpazolid (DZD)” NCT06114628
Known as LCB01-0371 “Delpazolid (LCB01-0371)” NCT05807399
7

NCT02882789

NCT03492996

NCT02529241

NCT02538003

NCT01554995

NCT01842516

NCT02540460

Modality Small molecule “LCB01-0371 is a novel oxazolidinone with broad-spectrum activity against Gram-positive pathogens in both in vitro studies and animal infection models.” PMID 29712654 Jun 2018
Route Oral “multiple oral dosing of LCB01-0371 (200-mg tablet or 400-mg tablet) for 7 days” PMID 30420289 Nov 2018