Drugs / Flonoltinib
last change Jul 2026 re-read 2 minutes ago

Flonoltinib

also known as Flonoltinib Maleate

targets CDK6, FLT3, JAK2 via inhibition

Developed for
myelofibrosis · acquired polycythemia vera · COVID-19
Investigated by
Chengdu Zenitar Biomedical Technology Co., Ltd

Trials 9 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 13 trials
Phase 1 NCT07612306 Jun → Oct 2026 expected Chengdu Zenitar Biomedical Technology Co., Ltd Not yet recruiting No outcome recorded
Phase 1 NCT06387966 Mar → Aug 2024 Chengdu Zenitar Biomedical Technology Co., Ltd Completed No outcome recorded
Phase 1 NCT05115344 Nov 2021 → Dec 2022 myelofibrosis Chengdu Zenitar Biomedical Technology Co., Ltd Unknown No outcome recorded
Phase 1/21 trial
Phase 1/2 NCT05153343 Dec 2021 → Nov 2023 myelofibrosis Chengdu Zenitar Biomedical Technology Co., Ltd Completed No outcome recorded
Phase 23 trials
Phase 2 NCT07443306 Mar 2026 → Dec 2027 expected Chengdu Zenitar Biomedical Technology Co., Ltd Recruiting No outcome recorded
Phase 2 NCT07232290 Sep 2025 → Jul 2027 expected acquired polycythemia vera Chengdu Zenitar Biomedical Technology Co., Ltd Recruiting No outcome recorded
Phase 2 NCT06457425 May 2024 → May 2026 overdue Chengdu Zenitar Biomedical Technology Co., Ltd Recruiting No outcome recorded
Phase 31 trial
Phase 3 NCT07317700 Feb 2026 → Dec 2027 expected Chengdu Zenitar Biomedical Technology Co., Ltd Recruiting No outcome recorded
Phase not applicable1 trial
NCT05713279 Jan → Nov 2023 COVID-19 Chengdu Zenitar Biomedical Technology Co., Ltd Unknown No outcome recorded

Evidence & citations 5 cited values

Every value below carries the sentence it was read from. 10 sources stand behind the page.

FieldValueCited text
Known as Flonoltinib “Study of Flonoltinib Maleate Tablets in the Treatment of Severe Novel Coronavirus (COVID-19) Infection” NCT05713279
8

NCT05153343

NCT07612306

NCT07232290

NCT07317700

NCT06457425

NCT05115344

NCT07443306

NCT06387966

Known as Flonoltinib Maleate Flonoltinib Maleate (FM), a triple target inhibitor of JAK2/FLT3/CDK6, has the potential to inhibit JAK2 signaling pathway activity and treat bone marrow proliferative tumors.” NCT07232290
4

Flonoltinib maleate (FM), a novel JAK2/FLT3/CDK6 inhibitor, shows preliminary potential in improving hematologic parameters and reducing fibrosis.” PMID 41883618 Mar 2026

Flonoltinib Maleate (FM) targets Janus kinase 2 (JAK2) and FMS-like tyrosine kinase 3 (FLT3).” NCT05115344

Flonoltinib Maleate (FM) targets Janus kinase 2 (JAK2) and FMS-like tyrosine kinase 3 (FLT3).” NCT05153343

“A Clinical Trial of Flonoltinib Maleate for Intermediate or High-Risk Myelofibrosis” NCT07317700

Action Inhibit “FM is a dual target inhibitor of JAK2/FLT3.” NCT05153343
Route Oral “single and repeated oral administration of flonoltinib maleate tablets” NCT05115344
Target JAK2 “FM targets Janus kinase 2 (JAK2)” NCT05153343