Drugs / voxtalisib
last change May 2018 re-read 2 minutes ago

voxtalisib

also known as SAR245409 · XL765

Small molecule targets MTOR via inhibition

Developed for
cancer · breast cancer · glioblastoma · non-small cell lung carcinoma · astrocytoma (excluding glioblastoma) · B-cell chronic lymphocytic leukemia · colorectal cancer · lymphoma
+5 more · mantle cell lymphoma · melanoma · metastatic neoplasm · mixed glioma · ovarian cancer
Investigated by
Sanofi · EMD Serono

Trials 11 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 17 trials
Phase 1 NCT01596270 Jun 2012 → Oct 2014 cancer Sanofi Completed No outcome recorded
Phase 1 NCT01410513 Dec 2011 → May 2014 B-cell chronic lymphocytic leukemia, mantle cell lymphoma Sanofi Completed No outcome recorded
Phase 1 NCT01390818 May 2011 → Apr 2015 breast cancer, colorectal cancer, melanoma, metastatic neoplasm +1 EMD Serono Completed No outcome recorded
Phase 1 NCT01240460 Jan 2011 → Jun 2012 astrocytoma (excluding glioblastoma), glioblastoma Sanofi Completed No outcome recorded
Phase 1 NCT00777699 Aug 2008 → Feb 2011 non-small cell lung carcinoma Sanofi Completed No outcome recorded
Phase 1 NCT00704080 Aug 2008 → Feb 2012 glioblastoma, mixed glioma Sanofi Completed No outcome recorded
Phase 1 NCT00485719 Jun 2007 → Sep 2012 cancer Sanofi Completed No outcome recorded
Phase 1/22 trials
Phase 1/2 NCT01587040 Jul 2012 → May 2018 cancer Sanofi Completed No outcome recorded
Phase 1/2 NCT01082068 Jun 2010 → Apr 2013 breast cancer Sanofi Completed No outcome recorded
Phase 22 trials
Phase 2 NCT01936363 Sep 2013 → May 2015 ovarian cancer EMD Serono Completed No outcome recorded
Phase 2 NCT01403636 Oct 2011 → Sep 2014 lymphoma Sanofi Completed No outcome recorded

Evidence & citations 7 cited values

Every value below carries the sentence it was read from. 13 sources stand behind the page.

FieldValueCited text
Known as voxtalisib “We aimed to investigate the efficacy and safety of voxtalisib (also known as XL765 or SAR245409), a pan-PI3K/mTOR inhibitor, in patients with relapsed or refractory lymphoma,...” PMID 29550382 Mar 2018
Known as SAR245409 “XL765 (SAR245409) is a dual PI3K and mTOR inhibitor.” NCT01240460
10

“XL765 (SAR245409)” NCT00485719

“XL765 (SAR245409)” NCT01082068

“XL765 (SAR245409)” NCT00777699

“XL765 (SAR245409)” NCT00704080

NCT01587040

NCT01936363

NCT01410513

NCT01403636

NCT01596270

NCT01390818

Known as XL765 “We aimed to investigate the efficacy and safety of voxtalisib (also known as XL765 or SAR245409), a pan-PI3K/mTOR inhibitor, in patients with relapsed or refractory lymphoma,...” PMID 29550382 Mar 2018
5

NCT00777699

NCT01240460

NCT00485719

NCT00704080

NCT01082068

Action Inhibit “XL765 is a new chemical entity that inhibits the kinases PI3K and mTOR” NCT00485719
Modality Small molecule “XL765 is a new chemical entity” NCT00777699
1

CHEMBL3545366

Route Oral “administered orally” NCT00485719
Target MTOR “XL765 is a new chemical entity that inhibits the kinases PI3K and mTOR.” NCT00777699