Drugs / vercirnon
last change Dec 2014 re-read 2 minutes ago

vercirnon

Small molecule targets CCR9 via inhibition

Developed for
Crohn disease · celiac disease · ulcerative colitis
Investigated by
GlaxoSmithKline · Amgen

Trials 11 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 14 trials
Phase 1 NCT01827631 May → Jun 2013 Crohn disease GlaxoSmithKline Completed No outcome recorded
Phase 1 NCT01489943 Sep → Nov 2011 Crohn disease GlaxoSmithKline Completed No outcome recorded
Phase 1 NCT01611805 Jul → Oct 2010 Crohn disease GlaxoSmithKline Completed No outcome recorded
Phase 1 NCT01114607 May → Jun 2010 Crohn disease GlaxoSmithKline Completed No outcome recorded
Phase 23 trials
Phase 2 NCT00540657 Oct 2007 → Jun 2008 celiac disease Amgen Completed No outcome recorded
Phase 2 NCT00306215 Mar 2006 → Aug 2008 Crohn disease Amgen Completed No outcome recorded
Phase 2 NCT00102921 Aug 2004 → Dec 2005 Crohn disease Amgen Completed No outcome recorded
Phase 34 trials
Phase 3 NCT01536418 Nov 2011 → Oct 2013 Crohn disease GlaxoSmithKline Terminated No outcome recorded
Phase 3 NCT01316939 May 2011 → Oct 2013 Crohn disease GlaxoSmithKline Terminated No outcome recorded
Phase 3 NCT01318993 Apr 2011 → Sep 2013 Crohn disease GlaxoSmithKline Terminated No outcome recorded
Phase 3 NCT01277666 Dec 2010 → Jul 2013 Crohn disease GlaxoSmithKline Completed No outcome recorded
Also used as a comparator or background therapy in 1 trial
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 2 NCT01658605 Comparator Feb 2013 ulcerative colitis GlaxoSmithKline Withdrawn No outcome recorded

Evidence & citations 11 cited values

Every value below carries the sentence it was read from. 14 sources stand behind the page.

FieldValueCited text
Known as vercirnon “CCX282-B, also called vercirnon, is a specific, orally-administered chemokine receptor CCR9 antagonist that regulates migration and activation of inflammatory cells in the intestine.” PMID 23527300 Mar 2013
Known as CCX282 ChEMBL registry synonym — accepted as the source's own label CHEMBL2178578
Known as CCX282-B ClinicalTrials.gov intervention name — accepted as the source's own label NCT00306215
2

NCT00102921

NCT00540657

Known as GSK1605786 ClinicalTrials.gov intervention name — accepted as the source's own label NCT01658605
4

NCT01827631

NCT01489943

NCT01611805

NCT01114607

Known as GSK1605786A ClinicalTrials.gov intervention name — accepted as the source's own label NCT01277666
3

NCT01536418

NCT01316939

NCT01318993

Known as VERCIRNON SODIUM ChEMBL registry synonym — accepted as the source's own label CHEMBL2178578
Known as Verecimon ChEMBL registry synonym — accepted as the source's own label CHEMBL2178578
Action Inhibit “CCX282-B is a highly potent, orally active, chemokine receptor antagonist” NCT00102921
Modality Small molecule CHEMBL2178578
Route Oral “daily oral doses of CCX282-B” NCT00102921
Target CCR9 “whose single target is the G-protein coupled receptor CCR9.” NCT00102921