Drugs / Basimglurant
last change Apr 2025 re-read 2 minutes ago

Basimglurant

Small molecule targets GRM5

Developed for
fragile X syndrome · major depressive disorder · depressive disorder · trigeminal neuralgia · tuberous sclerosis
Investigated by
Hoffmann-La Roche · Noema Pharma AG

Trials 15 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 18 trials
Phase 1 NCT02433093 Apr → Sep 2015 major depressive disorder Hoffmann-La Roche Completed No outcome recorded
Phase 1 NCT01873508 Jun → Aug 2013 Hoffmann-La Roche Completed No outcome recorded
Phase 1 NCT01665404 Jul → Sep 2012 Hoffmann-La Roche Completed No outcome recorded
Phase 1 NCT01629368 Jun → Sep 2012 Hoffmann-La Roche Completed No outcome recorded
Phase 1 NCT01592890 Apr → May 2012 Hoffmann-La Roche Completed No outcome recorded
Phase 1 NCT01483469 Dec 2011 → Oct 2013 Hoffmann-La Roche Completed No outcome recorded
Phase 1 NCT01368926 Jun → Nov 2011 Hoffmann-La Roche Completed No outcome recorded
Phase 1 NCT01045083 Jan 2010 → Jun 2011 Hoffmann-La Roche Completed No outcome recorded
Phase 26 trials
Phase 2 NCT05059327 Mar 2022 → Feb 2025 tuberous sclerosis Noema Pharma AG Completed No outcome recorded
Phase 2 NCT01750957 Feb 2013 → Apr 2014 fragile X syndrome Hoffmann-La Roche Completed No outcome recorded
Phase 2 NCT01517698 May 2012 → Apr 2014 fragile X syndrome Hoffmann-La Roche Completed No outcome recorded
Phase 2 NCT01437657 Oct 2011 → Sep 2013 major depressive disorder Hoffmann-La Roche Completed No outcome recorded
Phase 2 NCT01015430 Nov 2009 → Jan 2011 fragile X syndrome Hoffmann-La Roche Completed No outcome recorded
Phase 2 NCT00809562 Mar 2009 → Feb 2011 depressive disorder Hoffmann-La Roche Completed No outcome recorded
Phase 2/31 trial
Phase 2/3 NCT05217628 Jan 2022 → Feb 2027 expected trigeminal neuralgia Noema Pharma AG Active not recruiting No outcome recorded

Evidence & citations 10 cited values

Every value below carries the sentence it was read from. 16 sources stand behind the page.

FieldValueCited text
Known as Basimglurant “Efficacy and Safety of Basimglurant as Adjunctive Therapy for Major Depression:” PMID 27304433 Jul 2016
3

NCT05217628

NCT02433093

NCT05059327

Known as NOE-101 “The study drug (NOE-101, basimglurant) is a potent inhibitor of metabotropic glutamate receptor 5 (mGluR5)” NCT05059327
1

NOE-101NCT05217628

Known as RG-7090 ChEMBL registry synonym — accepted as the source's own label CHEMBL3301626
Known as RO4917523 ClinicalTrials.gov intervention name — accepted as the source's own label NCT01665404
10

NCT00809562

NCT01629368

NCT01517698

NCT01483469

NCT01750957

NCT01015430

NCT01045083

NCT01592890

NCT01368926

NCT01873508

Known as RO4917523-000 ChEMBL registry synonym — accepted as the source's own label CHEMBL3301626
Known as RO4917523-009 SULPHATE ChEMBL registry synonym — accepted as the source's own label CHEMBL3301626
Action Inhibit “Antagonism of the postsynaptic metabotropic glutamate subtype 5 receptor” PMID 27304433 Jul 2016
Modality Small molecule CHEMBL3301626
Route Oral “daily oral RO4917523” NCT00809562
Target GRM5 “Metabotropic glutamate receptor 5 modulator” CHEMBL3301626