Drugs / Odanacatib
last change Nov 2020 re-read 2 minutes ago

Odanacatib

also known as MK0822 · ODN · L-001037536 · L-1037536

Small molecule targets CTSK via inhibition

Developed for
osteoporosis · postmenopausal osteoporosis · breast cancer · metastatic carcinoma in the bone · osteoarthritis · prostate cancer
Investigated by
Merck Sharp & Dohme LLC

Trials 20 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 18 trials
Phase 1 NCT01630616 Mar 2013 → Jul 2016 osteoporosis Merck Sharp & Dohme LLC Terminated No outcome recorded
Phase 1 NCT01512693 Feb → Apr 2012 liver disorder Merck Sharp & Dohme LLC Completed No outcome recorded
Phase 1 NCT01512667 Jan → Aug 2012 impaired renal function disease Merck Sharp & Dohme LLC Completed No outcome recorded
Phase 1 NCT01068262 Dec 2009 → Apr 2010 osteoporosis Merck Sharp & Dohme LLC Completed No outcome recorded
Phase 1 NCT00863525 Nov → Dec 2004 osteoporosis Merck Sharp & Dohme LLC Completed No outcome recorded
Phase 1 NCT00770159 Nov 2004 → Jun 2005 osteoporosis Merck Sharp & Dohme LLC Completed No outcome recorded
Phase 1 NCT00769418 Sep → Dec 2004 osteoporosis Merck Sharp & Dohme LLC Completed No outcome recorded
Phase 1 NCT00863590 Jun 2004 → Feb 2005 osteoporosis Merck Sharp & Dohme LLC Completed No outcome recorded
Phase 25 trials
Phase 2 NCT00885170 Apr 2009 → Sep 2011 osteoporosis Merck Sharp & Dohme LLC Completed No outcome recorded
Phase 2 NCT00620113 Dec 2007 → May 2009 postmenopausal osteoporosis Merck Sharp & Dohme LLC Completed No outcome recorded
Phase 2 NCT00399802 Nov 2006 → Dec 2007 breast cancer, metastatic carcinoma in the bone Merck Sharp & Dohme LLC Completed No outcome recorded
Phase 2 NCT00397683 Oct 2006 → Apr 2007 osteoarthritis Merck Sharp & Dohme LLC Terminated No outcome recorded
Phase 2 NCT00112437 Jun 2005 → Dec 2007 osteoporosis Merck Sharp & Dohme LLC Completed No outcome recorded
Phase 37 trials
Phase 3 NCT01803607 Mar 2013 → Nov 2014 osteoporosis Merck Sharp & Dohme LLC Terminated No outcome recorded
Phase 3 NCT01552122 May 2012 → Feb 2015 postmenopausal osteoporosis Merck Sharp & Dohme LLC Withdrawn No outcome recorded
Phase 3 NCT01120600 Jun 2010 → Jul 2013 osteoporosis Merck Sharp & Dohme LLC Completed No outcome recorded
Phase 3 NCT00729183 Oct 2008 → Mar 2010 osteoporosis Merck Sharp & Dohme LLC Completed No outcome recorded
Phase 3 NCT00691899 Sep 2008 prostate cancer Merck Sharp & Dohme LLC Withdrawn No outcome recorded
Phase 3 NCT00692458 Sep 2008 breast cancer Merck Sharp & Dohme LLC Withdrawn No outcome recorded
Phase 3 NCT00529373 Sep 2007 → Nov 2012 postmenopausal osteoporosis Merck Sharp & Dohme LLC Terminated No outcome recorded

Evidence & citations 9 cited values

Every value below carries the sentence it was read from. 26 sources stand behind the page.

FieldValueCited text
Known as odanacatib ClinicalTrials.gov intervention name — accepted as the source's own label NCT00692458
16

NCT00769418

NCT00399802

NCT01552122

NCT00112437

NCT00863525

NCT00863590

NCT00729183

NCT00885170

NCT00620113

NCT01803607

NCT01068262

NCT00770159

NCT01630616

NCT01120600

NCT00691899

NCT00529373

Known as L-001037536 ChEMBL registry synonym — accepted as the source's own label CHEMBL481611
Known as L-1037536 ChEMBL registry synonym — accepted as the source's own label CHEMBL481611
Known as MK0822 “This study will assess the safety, tolerability, pharmacokinetics, and pharmacodynamics of once-daily multiple-dose administration of odanacatib (MK0822).” NCT00769418
5

“A Single-Dose Study of the Safety, Tolerability, and Pharmacokinetics of Odanacatib (MK0822) in Healthy Volunteers” NCT00863590

“Odanacatib (MK0822)” NCT00770159

NCT01512667

NCT00397683

NCT01512693

Known as ODN “Odanacatib (ODN) is a selective cathepsin K inhibitor being developed to treat osteoporosis.” PMID 24064689 Sep 2013
2

“Odanacatib (ODN) was investigated as an osteoporosis treatment in 292 men.” PMID 33200257 Nov 2020

“odanacatib (ODN), a cathepsin K inhibitor, in humans.” PMID 23013236 May 2013

Action Inhibit “Odanacatib selectively and reversibly inhibited cathepsin K” PMID 19874198 May 2010
Modality Small molecule CHEMBL481611
Route Oral “The efficacy and safety of weekly oral odanacatib (ODN) 50 mg for up to 8 years were assessed” PMID 26879200 Feb 2016
Target CTSK “Odanacatib (ODN) is a selective cathepsin K inhibitor being developed to treat osteoporosis.” PMID 24064689 Sep 2013