Drugs / Elironrasib
last change Jan 2026 re-read 2 minutes ago

Elironrasib

also known as RMC-6291

targets KRAS via inhibition

Developed for
non-small cell lung carcinoma · colorectal cancer · pancreatic ductal adenocarcinoma · colorectal carcinoma · metastatic neoplasm · lung cancer
Investigated by
Revolution Medicines, Inc. · Summit Therapeutics

Trials 4 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 11 trial
Phase 1 NCT05462717 Sep 2022 → Mar 2027 expected colorectal carcinoma, non-small cell lung carcinoma, pancreatic ductal adenocarcinoma Revolution Medicines, Inc. Active not recruiting No outcome recorded
Phase 1/23 trials
Phase 1/2 NCT07397338 Jan 2026 → May 2029 expected colorectal cancer, metastatic neoplasm, non-small cell lung carcinoma Revolution Medicines, Inc. Recruiting No outcome recorded
Phase 1/2 NCT06162221 Jan 2024 → Jun 2027 expected non-small cell lung carcinoma Revolution Medicines, Inc. Recruiting No outcome recorded
Phase 1/2 NCT06128551 Nov 2023 → Dec 2028 expected colorectal cancer, non-small cell lung carcinoma, pancreatic ductal adenocarcinoma Revolution Medicines, Inc. Recruiting No outcome recorded

Evidence & citations 6 cited values

Every value below carries the sentence it was read from. 5 sources stand behind the page.

FieldValueCited text
Known as Elironrasib ClinicalTrials.gov intervention name — accepted as the source's own label NCT06128551
1

NCT07397338

Known as RMC-6291 ClinicalTrials.gov intervention name — accepted as the source's own label NCT06162221
1

NCT05462717

Action Inhibit “RMC-6291 (KRAS G12C(ON) inhibitor)” NCT05462717
Modality Small molecule “We designed a natural product-inspired small molecule that remodels the surface of cyclophilin A (CYPA) to create a neomorphic interface with high affinity and selectivity for...” PMID 37590355 Aug 2023
Route Oral Oral tablet once or twice a day” NCT05462717
Target KRAS “RMC-6291 (KRAS G12C(ON) inhibitor)” NCT05462717