Drugs / Imgatuzumab
last change Aug 2022 re-read 2 minutes ago

Imgatuzumab

also known as RO5083945 · GA201 · HUMA-B · HuMAB<EGFR> · RG7160

Monoclonal antibody targets EGFR, FCGR3A

Developed for
non-small cell lung carcinoma · colorectal cancer · head and neck squamous cell carcinoma · neoplasm · skin squamous cell carcinoma
Investigated by
Hoffmann-La Roche · ICON plc · Pega-One S.A.S.

Trials 6 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 13 trials
Phase 1 NCT01702714 Jul 2014 → Feb 2016 non-small cell lung carcinoma Hoffmann-La Roche Withdrawn No outcome recorded
Phase 1 NCT01046266 Nov 2009 → Jun 2012 head and neck squamous cell carcinoma Hoffmann-La Roche Completed No outcome recorded
Phase 1 NCT00721266 Jun 2008 → Jun 2011 neoplasm Hoffmann-La Roche Completed No outcome recorded
Phase 23 trials
Phase 2 NCT04985825 Dec 2021 → Aug 2022 skin squamous cell carcinoma Pega-One S.A.S. Withdrawn No outcome recorded
Phase 2 NCT01326000 Apr 2011 → Dec 2013 colorectal cancer Hoffmann-La Roche Completed No outcome recorded
Phase 2 NCT01185847 Nov 2010 → Sep 2012 non-small cell lung carcinoma Hoffmann-La Roche Completed No outcome recorded

Evidence & citations 11 cited values

Every value below carries the sentence it was read from. 9 sources stand behind the page.

FieldValueCited text
Known as imgatuzumab “glycoengineered imgatuzumab (GA201; 700 or 1400 mg)” PMID 28950289 Nov 2017
1

NCT04985825

Known as GA201 “Phase I pharmacokinetic and pharmacodynamic dose-escalation study of RG7160 (GA201), the first glycoengineered monoclonal antibody against the epidermal growth factor receptor,...” PMID 21900113 Sep 2011
1

“glycoengineered imgatuzumab (GA201; 700 or 1400 mg)” PMID 28950289 Nov 2017

Known as HUMA-B ChEMBL registry synonym — accepted as the source's own label CHEMBL2109389
Known as HuMAB<EGFR> ChEMBL registry synonym — accepted as the source's own label CHEMBL2109389
Known as RG7160 “Phase I pharmacokinetic and pharmacodynamic dose-escalation study of RG7160 (GA201), the first glycoengineered monoclonal antibody against the epidermal growth factor receptor,...” PMID 21900113 Sep 2011
Known as RO5083945 ClinicalTrials.gov intervention name — accepted as the source's own label NCT01046266
4

NCT01326000

NCT01702714

NCT00721266

NCT01185847

Action Inhibit “anti-epidermal growth factor receptor (EGFR)” PMID 21900113 Sep 2011
Modality Monoclonal antibody “RG7160 (GA201), a humanized and glycoengineered immunoglobulin G(1) anti-epidermal growth factor receptor (EGFR) monoclonal antibody with enhanced antibody-dependent...” PMID 21900113 Sep 2011
Route Intravenous “Administered iv, either weekly, every 2 weeks or every 3 weeks” NCT00721266
Target EGFR “anti-epidermal growth factor receptor (EGFR) monoclonal antibody” PMID 21900113 Sep 2011
Target FCGR3A “Low affinity immunoglobulin gamma Fc region receptor III-A cross-linking agent” CHEMBL2109389