Drugs / DASOLAMPANEL ETIBUTIL
last change Jun 2010 re-read 2 minutes ago

DASOLAMPANEL ETIBUTIL

Small molecule targets GRM5 via inhibition

Developed for
diabetic neuropathy · osteoarthritis, knee
Investigated by
Eli Lilly and Company

Trials 2 · a red edge is where a trial was stopped

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PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 2 NCT00790790 Nov 2008 → Jan 2010 osteoarthritis, knee Eli Lilly and Company Completed No outcome recorded
Phase 2 NCT00785577 Nov 2008 → May 2010 diabetic neuropathy Eli Lilly and Company Completed No outcome recorded

Evidence & citations 7 cited values

Every value below carries the sentence it was read from. 3 sources stand behind the page.

FieldValueCited text
Known as DASOLAMPANEL ETIBUTIL ChEMBL registry synonym — accepted as the source's own label CHEMBL2107328
Known as DASOLAMPANEL ETIBUTIL TOSYLATE ChEMBL registry synonym — accepted as the source's own label CHEMBL2107328
Known as LY545694 ClinicalTrials.gov intervention name — accepted as the source's own label NCT00790790
1

NCT00785577

Action Inhibit “Metabotropic glutamate receptor 5 antagonist” CHEMBL2107328
1

“LY545694, an iGluR5 Antagonist” NCT00785577

Modality Small molecule CHEMBL2107328
Route Oral “LY545694 21 mg BID po for 1 week” NCT00785577
Target GRM5 “Metabotropic glutamate receptor 5 antagonist” CHEMBL2107328