Drugs / TAK-733
last change Feb 2025 re-read 2 minutes ago

TAK-733

also known as REC-4881 · Mek inhibitor tak-733

Small molecule targets MAP2K1, MAP2K2 via inhibition

Developed for
neoplasm · classic familial adenomatous polyposis · melanoma
Investigated by
Millennium Pharmaceuticals, Inc. · Recursion Pharmaceuticals Inc.

Trials 4 · a red edge is where a trial was stopped

201020112012201320142015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 12 trials
Phase 1 NCT01613261 Aug 2013 → Sep 2015 neoplasm Millennium Pharmaceuticals, Inc. Withdrawn No outcome recorded
Phase 1 NCT00948467 Dec 2009 → Apr 2013 melanoma Millennium Pharmaceuticals, Inc. Completed No outcome recorded
Phase 1/21 trial
Phase 1/2 NCT05552755 Jul 2023 → Jun 2027 expected classic familial adenomatous polyposis Recursion Pharmaceuticals Inc. Recruiting No outcome recorded
Phase 21 trial
Phase 2 NCT06005974 Jan 2024 → Feb 2025 neoplasm Recursion Pharmaceuticals Inc. Terminated No outcome recorded

Evidence & citations 8 cited values

Every value below carries the sentence it was read from. 5 sources stand behind the page.

FieldValueCited text
Known as TAK-733 ClinicalTrials.gov intervention name — accepted as the source's own label NCT01613261
1

NCT00948467

Known as Mek inhibitor tak-733 ChEMBL registry synonym — accepted as the source's own label CHEMBL1615025
Known as REC-4881 ClinicalTrials.gov intervention name — accepted as the source's own label NCT05552755
1

NCT06005974

Action Inhibit “Dual specificity mitogen-activated protein kinase kinase 1 inhibitor” CHEMBL1615025
2

“Dual specificity mitogen-activated protein kinase kinase 2 inhibitor” CHEMBL1615025

“an Oral MEK Inhibitor” NCT00948467

Modality Small molecule “an Oral MEK Inhibitor” NCT00948467
1

CHEMBL1615025

Route Oral “TAK-733 will be administered orally” NCT00948467
Target MAP2K1 “Dual specificity mitogen-activated protein kinase kinase 1 inhibitor” CHEMBL1615025
Target MAP2K2 “Dual specificity mitogen-activated protein kinase kinase 2 inhibitor” CHEMBL1615025