Drugs / vabicaserin
last change Sep 2009 re-read 2 minutes ago

vabicaserin

Small molecule targets HTR2A, HTR2B, HTR2C via inhibition / activation

Developed for
schizophrenia
Investigated by
Wyeth is now a wholly owned subsidiary of Pfizer · Pfizer

Trials 9 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 16 trials
Phase 1 NCT00928551 Jun → Sep 2009 Wyeth is now a wholly owned subsidiary of Pfizer Completed No outcome recorded
Phase 1 NCT00541996 Aug → Oct 2007 schizophrenia Wyeth is now a wholly owned subsidiary of Pfizer Completed No outcome recorded
Phase 1 NCT00505973 Jul → Oct 2007 schizophrenia Wyeth is now a wholly owned subsidiary of Pfizer Completed No outcome recorded
Phase 1 NCT00458107 Apr → Sep 2007 schizophrenia Wyeth is now a wholly owned subsidiary of Pfizer Completed No outcome recorded
Phase 1 NCT00420706 Dec 2006 Wyeth is now a wholly owned subsidiary of Pfizer Terminated No outcome recorded
Phase 1 NCT00447941 Jun → Aug 2006 schizophrenia Wyeth is now a wholly owned subsidiary of Pfizer Completed No outcome recorded
Phase 23 trials
Phase 2 NCT00768612 Nov 2008 → Jul 2009 schizophrenia Wyeth is now a wholly owned subsidiary of Pfizer Withdrawn No outcome recorded
Phase 2 NCT00563706 Dec 2007 → Jun 2008 schizophrenia Pfizer Completed No outcome recorded
Phase 2 NCT00265551 Jan 2006 → Jan 2007 schizophrenia Wyeth is now a wholly owned subsidiary of Pfizer Completed No outcome recorded

Evidence & citations 12 cited values

Every value below carries the sentence it was read from. 10 sources stand behind the page.

FieldValueCited text
Known as vabicaserin “A Randomized, Double-Blind, Risperidone-Reference, Parallel-Group, Safety, and Tolerability Study of Vabicaserin (SCA-136) in Japanese Subjects With Acute Exacerbation of Schizophrenia” NCT00768612
3

NCT00928551

NCT00541996

NCT00563706

Known as SCA-136 “A Randomized, Open-Label, Single-Dose, 4-Period Crossover, Comparative Bioavailability Study of 3 Sustained- Release Formulations and an Immediate- Release Formulation of...” NCT00541996
7

“The primary purpose of this protocol is to establish the efficacy, safety, and tolerability of vabicaserin (SCA-136) using a once a day capsule in subjects with acute...” NCT00563706

“A Randomized, Double-Blind, Risperidone-Reference, Parallel-Group, Safety, and Tolerability Study of Vabicaserin (SCA-136) in Japanese Subjects With Acute Exacerbation of Schizophrenia” NCT00768612

NCT00265551

NCT00447941

NCT00420706

NCT00505973

NCT00458107

Known as VABICASERIN HYDROCHLORIDE ChEMBL registry synonym — accepted as the source's own label CHEMBL2110670
Known as Vabicaserina ChEMBL registry synonym — accepted as the source's own label CHEMBL2110670
Known as Vabicaserine ChEMBL registry synonym — accepted as the source's own label CHEMBL2110670
Action Activate “Serotonin 2c (5-HT2c) receptor agonist” CHEMBL2110670
Action Inhibit “Serotonin 2a (5-HT2a) receptor antagonist” CHEMBL2110670
1

“Serotonin 2b (5-HT2b) receptor antagonist” CHEMBL2110670

Modality Small molecule CHEMBL2110670
Route Oral “Administered Orally” NCT00447941
Target HTR2A “Serotonin 2a (5-HT2a) receptor antagonist” CHEMBL2110670
Target HTR2B “Serotonin 2b (5-HT2b) receptor antagonist” CHEMBL2110670
Target HTR2C “Serotonin 2c (5-HT2c) receptor agonist” CHEMBL2110670