Drugs / naratriptan
last change Jun 2020 re-read 2 minutes ago

naratriptan

Small molecule targets HTR1B, HTR1D via activation

Developed for
antisocial personality disorder · intermittent explosive disorder · migraine disorder · psychotic disorder

Regulatory milestones approvals, filings & regulatory actions · 1 recorded

MilestoneJurisdictionBrandIndicationDateSentence it was read from
Approved US (FDA) AMERGE 1998-02-10 fda.gov

Trials 0

Also used as a comparator or background therapy in 6 trials
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1/21 trial
Phase 1/2 NCT03066544 Comparator Nov 2016 → Dec 2019 migraine disorder Hartford HealthCare Unknown No outcome recorded
Phase 32 trials
Phase 3 NCT01726920 Comparator Jul → Dec 2014 migraine disorder Ache Laboratorios Farmaceuticos S.A. Withdrawn No outcome recorded
Phase 3 NCT01390324 Comparator Dec 2011 → Mar 2012 migraine disorder Ache Laboratorios Farmaceuticos S.A. Withdrawn No outcome recorded
Phase 43 trials
Phase 4 NCT01086358 Comparator Sep 2009 → Aug 2016 The Cleveland Clinic Completed No outcome recorded
Phase 4 NCT00282165 Comparator Nov 2006 → Dec 2012 antisocial personality disorder, intermittent explosive disorder, psychotic disorder UMC Utrecht Terminated No outcome recorded
Phase 4 NCT00487578 Comparator Oct 2006 → Oct 2009 Cady, Roger, M.D. Terminated No outcome recorded

Evidence & citations 11 cited values

Every value below carries the sentence it was read from. 7 sources stand behind the page.

FieldValueCited text
Known as naratriptan “Usual prescribed triptans may include:sumatriptan, rizatriptan, naratriptan, almotriptan, eletriptan, zolmitriptan” NCT01086358
5

NCT01726920

NCT00487578

NCT00282165

NCT01390324

NCT03066544

Known as Amerge ChEMBL registry synonym — accepted as the source's own label CHEMBL1278
Known as GR 85548A ChEMBL registry synonym — accepted as the source's own label CHEMBL1278
Known as Naramig ChEMBL registry synonym — accepted as the source's own label CHEMBL1278
Known as naratriptan HCl “Drug: naratriptan HClNCT00487578
Known as NARATRIPTAN HYDROCHLORIDE ChEMBL registry synonym — accepted as the source's own label CHEMBL1278
Action Activate “Serotonin 1d (5-HT1d) receptor agonist” CHEMBL1278
1

“Serotonin 1b (5-HT1b) receptor agonist” CHEMBL1278

Modality Small molecule CHEMBL1278
Route Oral “four weeks double blind experimental treatment using oral naratriptan” NCT00282165
Target HTR1B “Serotonin 1b (5-HT1b) receptor agonist” CHEMBL1278
Target HTR1D “Serotonin 1d (5-HT1d) receptor agonist” CHEMBL1278