Drugs / Foliglurax
last change May 2020 re-read 2 minutes ago

Foliglurax

also known as PXT002331 · DT-1687 · Lu AF99757

Small molecule targets GRM4 via activation

Developed for
Parkinson disease
Investigated by
H. Lundbeck A/S · Prexton Therapeutics

Trials 7 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 15 trials
Phase 1 NCT04275115 Feb → Apr 2020 H. Lundbeck A/S Completed No outcome recorded
Phase 1 NCT04322227 Jan → May 2020 Parkinson disease H. Lundbeck A/S Terminated No outcome recorded
Phase 1 NCT04175132 Nov 2019 → Mar 2020 Parkinson disease H. Lundbeck A/S Terminated No outcome recorded
Phase 1 NCT04002895 Jun → Aug 2019 H. Lundbeck A/S Completed No outcome recorded
Phase 1 NCT02639221 Jan → Aug 2016 Parkinson disease Prexton Therapeutics Completed No outcome recorded
Phase 22 trials
Phase 2 NCT03331848 Jan 2018 → Feb 2019 Parkinson disease Prexton Therapeutics Withdrawn No outcome recorded
Phase 2 NCT03162874 Jul 2017 → Feb 2020 Parkinson disease Prexton Therapeutics Completed No outcome recorded

Evidence & citations 8 cited values

Every value below carries the sentence it was read from. 8 sources stand behind the page.

FieldValueCited text
Known as Foliglurax “Study to Evaluate the Efficacy, Safety and Tolerability of PXT002331 (Foliglurax) in Reducing Motor Complications of Levodopa Therapy in Parkinson Disease's Patients” NCT03162874
5

“PXT002331 (Foliglurax)” NCT03331848

NCT04175132

NCT04002895

NCT04322227

NCT04275115

Known as DT-1687 ChEMBL registry synonym — accepted as the source's own label CHEMBL4089083
Known as Lu AF99757 “Interventional, Open-label, Single-dose Study Investigating the Absorption, Metabolism and Excretion (AME) of Foliglurax (Lu AF99757) Following Oral Dosing of 14C-foliglurax to...” NCT04002895
Known as PXT002331 ClinicalTrials.gov intervention name — accepted as the source's own label NCT03162874
2

NCT02639221

NCT03331848

Action Activate “Metabotropic glutamate receptor 4 positive allosteric modulator” CHEMBL4089083
Modality Small molecule CHEMBL4089083
Route Oral “PXT002331 is administered orally as single and multiple doses” NCT02639221
Target GRM4 “Metabotropic glutamate receptor 4 positive allosteric modulator” CHEMBL4089083