Drugs / Vorbipiprant
last change May 2026 re-read 2 minutes ago

Vorbipiprant

Small molecule targets PTGER4 via inhibition

Developed for
colorectal cancer · colorectal carcinoma · gastric cancer
Investigated by
Rottapharm Biotech · Agenus Inc. · Gruppo Oncologico del Nord-Ovest

Trials 3 · a red edge is where a trial was stopped

2018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1/21 trial
Phase 1/2 NCT05205330 Nov 2021 → Dec 2026 expected colorectal cancer, gastric cancer Rottapharm Biotech Active not recruiting No outcome recorded
Phase 22 trials
Phase 2 NCT05845450 May 2023 → May 2026 overdue colorectal carcinoma Gruppo Oncologico del Nord-Ovest Recruiting No outcome recorded
Phase 2 NCT03163966 Oct 2017 → Jan 2019 Rottapharm Biotech Completed No outcome recorded

Evidence & citations 8 cited values

Every value below carries the sentence it was read from. 4 sources stand behind the page.

FieldValueCited text
Known as vorbipiprant “CR6086 (Vorbipiprant) is a potent and selective, orally bioavailable, targeted immunomodulator small molecule acting as an EP4 receptor antagonist.” NCT05205330
1

NCT05845450

Known as CR6086 ClinicalTrials.gov intervention name — accepted as the source's own label NCT05205330
1

NCT03163966

Known as CR6086 SODIUM SALT ChEMBL registry synonym — accepted as the source's own label CHEMBL6067994
Known as VORBIPIPRANT SODIUM ChEMBL registry synonym — accepted as the source's own label CHEMBL6067994
Action Inhibit “Prostanoid EP4 receptor antagonist” CHEMBL6067994
1

“EP4 receptor antagonist” NCT03163966

Modality Small molecule small molecule prostaglandin EP4 receptor antagonist” NCT03163966
Route Oral oral CR6086 capsules” NCT03163966
Target PTGER4 “Prostanoid EP4 receptor antagonist” CHEMBL6067994