Drugs / Muraglitazar
last change Apr 2009 re-read 2 minutes ago

Muraglitazar

Small molecule targets PPARA, PPARG via activation

Developed for
type 2 diabetes mellitus · diabetes mellitus · hyperlipidemia
Investigated by
Bristol-Myers Squibb · Merck Sharp & Dohme LLC

Trials 10 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 2/32 trials
Phase 2/3 NCT00240383 May 2002 → Jun 2006 type 2 diabetes mellitus Bristol-Myers Squibb Completed No outcome recorded
Phase 2/3 NCT00245388 Apr → Jul 2002 hyperlipidemia Bristol-Myers Squibb Completed No outcome recorded
Phase 38 trials
Phase 3 NCT00130806 Sep → Nov 2005 type 2 diabetes mellitus Merck Sharp & Dohme LLC Terminated No outcome recorded
Phase 3 NCT00106808 Aug 2005 → Aug 2006 type 2 diabetes mellitus Bristol-Myers Squibb Completed No outcome recorded
Phase 3 NCT00094991 May 2004 → May 2006 type 2 diabetes mellitus Bristol-Myers Squibb Completed No outcome recorded
Phase 3 NCT00095030 Feb 2004 → Mar 2006 type 2 diabetes mellitus Bristol-Myers Squibb Completed No outcome recorded
Phase 3 NCT00240370 Oct 2003 → Mar 2005 type 2 diabetes mellitus Bristol-Myers Squibb Completed No outcome recorded
Phase 3 NCT00162175 Jul 2003 → Nov 2005 diabetes mellitus Bristol-Myers Squibb Completed No outcome recorded
Phase 3 NCT00162240 Jun 2003 → May 2004 diabetes mellitus Bristol-Myers Squibb Completed No outcome recorded
Phase 3 NCT00246987 Jun 2003 → Apr 2004 type 2 diabetes mellitus Bristol-Myers Squibb Completed No outcome recorded

Evidence & citations 9 cited values

Every value below carries the sentence it was read from. 12 sources stand behind the page.

FieldValueCited text
Known as Muraglitazar ClinicalTrials.gov intervention name — accepted as the source's own label NCT00245388
9

NCT00095030

NCT00240383

NCT00246987

NCT00094991

NCT00130806

NCT00162240

NCT00240370

NCT00162175

NCT00106808

Known as BMS-298585-01 ChEMBL registry synonym — accepted as the source's own label CHEMBL186179
Known as BMS298585 “A Study to Assess the Efficacy and Tolerability of MK0478 (Muraglitazar, Also, BMS 298585) Coadministered With Insulin in Patients With Type 2 Diabetes” NCT00130806
2

“Mechanism of Action and Efficacy of Muraglitazar (BMS298585) in the Treatment of Type 2 Diabetic Patients” NCT00094991

“BMS-298585 (muraglitazar) alone in combination with pravastatin” NCT00245388

Known as MK0478 MK0478 (muraglitazar)” NCT00130806
Known as MURAGLITAZAR CHLORIDE ChEMBL registry synonym — accepted as the source's own label CHEMBL186179
Action Activate “a dual (alpha/gamma) peroxisome proliferator-activated receptor activator” PMID 20368202 Apr 2009
2

“Peroxisome proliferator-activated receptor gamma agonist” CHEMBL186179

“Peroxisome proliferator-activated receptor alpha agonist” CHEMBL186179

Modality Small molecule CHEMBL186179
Target PPARA “Peroxisome proliferator-activated receptor alpha agonist” CHEMBL186179
Target PPARG “Peroxisome proliferator-activated receptor gamma agonist” CHEMBL186179