Drugs / GW501516
last change Aug 2011 re-read 3 minutes ago

GW501516

also known as Cardarine · GSK-516 · GW-1516

Small molecule targets PPARD via activation

Developed for
hyperlipidemia · lip disorder · obesity disorder
Investigated by
GlaxoSmithKline

Trials 1

200420052006200720082009201020112012201320142015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 21 trial
Phase 2 NCT00158899 Aug 2004 → Jun 2006 hyperlipidemia GlaxoSmithKline Completed No outcome recorded
Comparator or background therapy1 trial
Phase 4 NCT00841217 Comparator Apr 2003 → Aug 2005 cardiovascular disorder, lip disorder, obesity disorder The University of Western Australia Completed No outcome recorded

Evidence & citations 8 cited values

Every value below carries the sentence it was read from. 4 sources stand behind the page.

FieldValueCited text
Known as GW501516 ClinicalTrials.gov intervention name — accepted as the source's own label NCT00158899 ↗
1

NCT00841217 ↗

Known as Cardarine ChEMBL registry synonym — accepted as the source's own label CHEMBL38943 ↗
Known as GSK-516 ChEMBL registry synonym — accepted as the source's own label CHEMBL38943 ↗
Known as GW-1516 ChEMBL registry synonym — accepted as the source's own label CHEMBL38943 ↗
Action Activate “GW501516, a PPAR-δ agonist” PMID 21816786 ↗ Aug 2011
Modality Small molecule — CHEMBL38943 ↗
Route Oral “GW501516 oral tablets” NCT00158899 ↗
Target PPARD “GW501516, a PPAR-δ agonist” PMID 21816786 ↗ Aug 2011