Drugs / Rivipansel
last change Nov 2019 re-read 2 minutes ago

Rivipansel

Small molecule targets SELE, SELL, SELP via inhibition

Developed for
sickle cell disease
Investigated by
GlycoMimetics Incorporated · Biossil Inc.

Trials 9 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 15 trials
Phase 1 NCT02998099 Jan → Feb 2017 GlycoMimetics Incorporated Completed No outcome recorded
Phase 1 NCT02871570 Sep 2016 → Feb 2017 GlycoMimetics Incorporated Completed No outcome recorded
Phase 1 NCT02813798 Jun 2016 → Feb 2018 impaired renal function disease GlycoMimetics Incorporated Completed No outcome recorded
Phase 1 NCT02217917 Oct 2015 → Apr 2016 GlycoMimetics Incorporated Completed No outcome recorded
Phase 1 NCT01941511 Aug 2013 → Aug 2014 GlycoMimetics Incorporated Completed No outcome recorded
Phase 1/21 trial
Phase 1/2 NCT00911495 May 2009 → Jul 2010 sickle cell disease GlycoMimetics Incorporated Completed No outcome recorded
Phase 21 trial
Phase 2 NCT01119833 May 2010 → Dec 2012 sickle cell disease GlycoMimetics Incorporated Completed No outcome recorded
Phase 32 trials
Phase 3 NCT02433158 Dec 2015 → Nov 2019 sickle cell disease GlycoMimetics Incorporated Terminated No outcome recorded
Phase 3 NCT02187003 Jun 2015 → May 2019 sickle cell disease Biossil Inc. Completed No outcome recorded

Press releases naming this drug 2 releases

DateIssuerRelease
2019-08-02 Pfizer Pfizer Announces Phase 3 Top-Line Results for Rivipansel in Patients with Sickle Cell Disease Experiencing a Vaso-Occlusive Crisis pfizer.com
2015-10-29 Pfizer GLYCOMIMETICS, INC. ANNOUNCES INITIATION OF FIRST CLINICAL TRIAL EVALUATING SUBCUTANEOUS ADMINISTRATION OF RIVIPANSEL pfizer.com

Evidence & citations 11 cited values

Every value below carries the sentence it was read from. 12 sources stand behind the page.

FieldValueCited text
Known as rivipansel “These results support a phase 3 study of GMI-1070 (now rivipansel) for SCD VOC.” PMID 25733584 Mar 2015
7

NCT02813798

NCT01941511

NCT02998099

NCT02433158

NCT02871570

NCT02217917

NCT02187003

Known as GMI 1070 “We performed a Phase 1 study of the selectin inhibitor GMI 1070 in patients with sickle cell anemia.” PMID 24988449 Jul 2014
2

NCT01119833

NCT00911495

Known as pf 06460031 “A Phase 1, Randomized, Double Blind, Sponsor Open, Placebo Controlled, Single And Multiple Ascending Dose Study To Evaluate The Safety, Tolerability, And Pharmacokinetics Of...” NCT02217917
Known as PF-06460031-02 ChEMBL registry synonym — accepted as the source's own label CHEMBL3707446
Known as RIVIPANSEL SODIUM ChEMBL registry synonym — accepted as the source's own label CHEMBL3707446
Action Inhibit “This Phase 1/Phase 2 study will evaluate GMI-1070, a pan-selectin inhibitor” NCT00911495
3

“Leukocyte adhesion molecule-1 antagonist” CHEMBL3707446

“Selectin E antagonist” CHEMBL3707446

“P-selectin antagonist” CHEMBL3707446

Modality Small molecule CHEMBL3707446
Route Intravenous Intravenous GMI-1070 given as two doses over the course of one day” NCT00911495
Target SELE Selectin E antagonist” CHEMBL3707446
Target SELL “Leukocyte adhesion molecule-1 antagonist” CHEMBL3707446
Target SELP “P-selectin antagonist” CHEMBL3707446