Drugs / CTP-499

Trials 4 · a red edge is where a trial was stopped

2012201320142015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 12 trials
Phase 1 NCT03836222 Feb → Jun 2018 Processa Pharmaceuticals Completed No outcome recorded
Phase 1 NCT01460199 Aug → Dec 2011 chronic kidney disease Concert Pharmaceuticals Completed No outcome recorded
Phase 22 trials
Phase 2 NCT04800562 Apr 2021 → Feb 2023 necrobiosis lipoidica Processa Pharmaceuticals Terminated No outcome recorded
Phase 2 NCT03698864 Nov 2018 → Feb 2020 necrobiosis lipoidica Processa Pharmaceuticals Completed No outcome recorded
Also used as a comparator or background therapy in 2 trials
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 11 trial
Phase 1 NCT01328821 Comparator Mar → Apr 2011 diabetic kidney disease Concert Pharmaceuticals Completed No outcome recorded
Phase 21 trial
Phase 2 NCT01487109 Comparator Jan 2012 → Jan 2015 chronic kidney disease, type 2 diabetes mellitus Concert Pharmaceuticals Completed No outcome recorded

Evidence & citations 6 cited values

Every value below carries the sentence it was read from. 8 sources stand behind the page.

FieldValueCited text
Known as CTP-499 ClinicalTrials.gov intervention name — accepted as the source's own label NCT01487109
2

NCT01328821

NCT01460199

Known as Deuterated s-lisofylline ChEMBL registry synonym — accepted as the source's own label CHEMBL4300766
Known as Lisophylline, (s)- ChEMBL registry synonym — accepted as the source's own label CHEMBL4300766
Known as PCS499 ClinicalTrials.gov intervention name — accepted as the source's own label NCT03836222
2

NCT03698864

NCT04800562

Modality Small molecule “PCS499, an oral deuterated pentoxifylline analog, may offer therapeutic benefit.” PMID 42054009 Jun 2026
1

CHEMBL4300766

Route Oral “PCS499, 900 mg, orally twice daily for 6 months, with optional 6-month extension.” PMID 42054009 Jun 2026