Drugs / Rineterkib
last change Sep 2024 re-read 2 minutes ago

Rineterkib

also known as LTT462

Small molecule

Developed for
melanoma · non-small cell lung carcinoma · colorectal cancer · myelofibrosis · ovarian neoplasm
Investigated by
Novartis Pharmaceuticals

Trials 5 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 13 trials
Phase 1 NCT04294160 Jul 2020 → Sep 2024 colorectal cancer Novartis Pharmaceuticals Terminated No outcome recorded
Phase 1 NCT02974725 Feb 2017 → Apr 2024 melanoma, non-small cell lung carcinoma Novartis Pharmaceuticals Terminated No outcome recorded
Phase 1 NCT02711345 Apr 2016 → Nov 2018 melanoma, non-small cell lung carcinoma, ovarian neoplasm Novartis Pharmaceuticals Terminated No outcome recorded
Phase 1/21 trial
Phase 1/2 NCT04097821 Sep 2019 → May 2023 myelofibrosis Novartis Pharmaceuticals Terminated No outcome recorded
Phase 21 trial
Phase 2 NCT04417621 Oct 2020 → Feb 2027 expected melanoma Novartis Pharmaceuticals Active not recruiting No outcome recorded

Evidence & citations 5 cited values

Every value below carries the sentence it was read from. 7 sources stand behind the page.

FieldValueCited text
Known as rineterkib “BACKGROUND: Genetic alterations activating the MAPK pathway are common in non-small cell lung cancer (NSCLC). Patients with NSCLC may benefit from treatment with the pan-RAF...” PMID 39383771 Sep 2024
1

NCT04097821

Known as LTT462 ClinicalTrials.gov intervention name — accepted as the source's own label NCT04417621
3

NCT02974725

NCT04294160

NCT02711345

Action Inhibit “ERK Inhibitor” NCT02711345
Modality Small molecule CHEMBL3909517
Route Oral “A Phase I Dose Finding Study of Oral LTT462 in Adult Patients With Advanced Solid Tumors Harboring MAPK Pathway Alterations.” NCT02711345