Drugs / GSK2816126
last change Jun 2017 re-read 3 minutes ago

GSK2816126

Small molecule targets EZH2 via inhibition

Developed for
cancer
Investigated by
GlaxoSmithKline

Trials 1

20142015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1 NCT02082977 Apr 2014 → Jun 2017 cancer GlaxoSmithKline Terminated No outcome recorded

Evidence & citations 5 cited values

Every value below carries the sentence it was read from. 2 sources stand behind the page.

FieldValueCited text
Known as GSK2816126 ClinicalTrials.gov intervention name — accepted as the source's own label NCT02082977 ↗
Action Inhibit “Histone-lysine N-methyltransferase EZH2 inhibitor” CHEMBL3287735 ↗
Modality Small molecule — CHEMBL3287735 ↗
Route Intravenous “given twice weekly by intravenous (IV) infusion.” NCT02082977 ↗
Target EZH2 “Histone-lysine N-methyltransferase EZH2 inhibitor” CHEMBL3287735 ↗