Drugs / ABT-639
last change Nov 2015 re-read 2 minutes ago

ABT-639

also known as Abt-639 free base

Small molecule targets CACNA1H via inhibition

Developed for
diabetic polyneuropathy
Investigated by
AbbVie

Trials 2 · a red edge is where a trial was stopped

20112012201320142015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 2 NCT01589432 Apr → Nov 2012 diabetic polyneuropathy AbbVie Completed No outcome recorded
Phase 2 NCT01345045 Apr → Oct 2011 diabetic polyneuropathy AbbVie Completed No outcome recorded

Evidence & citations 6 cited values

Every value below carries the sentence it was read from. 5 sources stand behind the page.

FieldValueCited text
Known as ABT-639 ClinicalTrials.gov intervention name — accepted as the source's own label NCT01345045
1

NCT01589432

Known as Abt-639 free base ChEMBL registry synonym — accepted as the source's own label CHEMBL3590674
Action Inhibit “a peripherally acting highly selective T-type Cav3.2 calcium channel blocker” PMID 26067585 Oct 2015
1

“Voltage-gated T-type calcium channel alpha-1H subunit blocker” CHEMBL3590674

Modality Small molecule CHEMBL3590674
Route Oral “single 100-mg oral dose of ABT-639” PMID 26035253 Nov 2015
Target CACNA1H “Voltage-gated T-type calcium channel alpha-1H subunit blocker” CHEMBL3590674