Drugs / GSK189254
last change Jan 2008 re-read 2 minutes ago

GSK189254

also known as [11C]GSK-189254

Small molecule targets HRH3 via inhibition

Developed for
narcolepsy
Investigated by
GlaxoSmithKline

Trials 2 · a red edge is where a trial was stopped

200720082009201020112012201320142015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 11 trial
Phase 1 NCT00387413 Oct 2006 → May 2007 GlaxoSmithKline Completed No outcome recorded
Phase 21 trial
Phase 2 NCT00366080 Nov 2006 → Jan 2008 narcolepsy GlaxoSmithKline Terminated No outcome recorded

Evidence & citations 6 cited values

Every value below carries the sentence it was read from. 3 sources stand behind the page.

FieldValueCited text
Known as GSK189254 ClinicalTrials.gov intervention name — accepted as the source's own label NCT00387413
1

NCT00366080

Known as [11C]GSK-189254 ChEMBL registry synonym — accepted as the source's own label CHEMBL517140
Action Inhibit “the Histamine H3 antagonist GSK189254” NCT00366080
1

“Histamine H3 receptor antagonist” CHEMBL517140

Modality Small molecule CHEMBL517140
Route Oral “The effects of repeated oral dosing of GSK189254 and duloxetine on secondary hyperalgesia in the EH model will be determined.” NCT00387413
Target HRH3 “Histamine H3 receptor antagonist” CHEMBL517140