Drugs / PREXIGEBERSEN
last change May 2020 re-read 2 minutes ago

PREXIGEBERSEN

Antisense oligonucleotide targets GRB2 via inhibition

Developed for
acute myeloid leukemia · myelodysplastic syndrome · Philadelphia-positive myelogenous leukemia · acute lymphoblastic leukemia
Investigated by
Bio-Path Holdings, Inc.

Trials 3 · a red edge is where a trial was stopped

2010201120122013201420152016201720182019202020212022202320242025202620272028
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 11 trial
Phase 1 NCT01159028 Jun 2010 → Mar 2017 Philadelphia-positive myelogenous leukemia, acute lymphoblastic leukemia, acute myeloid leukemia, myelodysplastic syndrome Bio-Path Holdings, Inc. Completed No outcome recorded
Phase 1/21 trial
Phase 1/2 NCT02923986 Sep 2017 → May 2020 Philadelphia-positive myelogenous leukemia, acute myeloid leukemia, myelodysplastic syndrome Bio-Path Holdings, Inc. Withdrawn No outcome recorded
Phase 21 trial
Phase 2 NCT02781883 May 2016 → Dec 2027 expected acute myeloid leukemia Bio-Path Holdings, Inc. Recruiting No outcome recorded

Evidence & citations 9 cited values

Every value below carries the sentence it was read from. 4 sources stand behind the page.

FieldValueCited text
Known as PREXIGEBERSEN ChEMBL registry synonym — accepted as the source's own label CHEMBL3989978
Known as BP-100-1.01/L-Grb2 ChEMBL registry synonym — accepted as the source's own label CHEMBL3989978
Known as BP1001 ClinicalTrials.gov intervention name — accepted as the source's own label NCT02781883
2

NCT02923986

NCT01159028

Known as L-grb-2 antisense ChEMBL registry synonym — accepted as the source's own label CHEMBL3989978
Known as L-Grb2 AS “The first goal of this clinical research study is to find the highest safe dose of BP1001, a liposomal Growth Factor Receptor Bound Protein-2 antisense oligodeoxynucleotide...” NCT01159028
Action Inhibit inhibit the cells from making Grb-2” NCT01159028
Modality Antisense oligonucleotide “antisense oligodeoxynucleotide” NCT01159028
Route Intravenous “administered by IV on twice weekly for 28 days” NCT01159028
Target GRB2 “inhibit the cells from making Grb-2” NCT01159028