Drugs / JI-101
last change Aug 2012 re-read 2 minutes ago

JI-101

Small molecule targets EPHB4, KDR, PDGFRB via inhibition

Developed for
cancer · colorectal cancer · neuroendocrine neoplasm · ovarian cancer
Investigated by
Jubilant Innovation Ltd. · University of Utah

Trials 2 · a red edge is where a trial was stopped

2009201020112012201320142015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1/2 NCT01149434 Sep 2010 → Aug 2012 colorectal cancer, neuroendocrine neoplasm, ovarian cancer University of Utah Terminated No outcome recorded
Phase 1/2 NCT00842335 Feb 2009 → Jul 2010 cancer Jubilant Innovation Ltd. Completed No outcome recorded

Evidence & citations 9 cited values

Every value below carries the sentence it was read from. 3 sources stand behind the page.

FieldValueCited text
Known as JI-101 ClinicalTrials.gov intervention name — accepted as the source's own label NCT00842335
1

NCT01149434

Known as Angiogenesis inhibitor ji-101 ChEMBL registry synonym — accepted as the source's own label CHEMBL3545155
Known as CGI-1842 ChEMBL registry synonym — accepted as the source's own label CHEMBL3545155
Action Inhibit “JI-101 is an inhibitor of vascular endothelial growth factor receptor 2 (VEGFR2), platelet-derived growth factor receptor beta (PDGFRβ), and EphB4 receptor” NCT00842335
3

“Vascular endothelial growth factor receptor 2 inhibitor” CHEMBL3545155

“Platelet-derived growth factor receptor beta inhibitor” CHEMBL3545155

“Ephrin type-B receptor 4 inhibitor” CHEMBL3545155

Modality Small molecule CHEMBL3545155
Route Oral “when given orally” NCT00842335
Target EPHB4 “Ephrin type-B receptor 4 inhibitor” CHEMBL3545155
Target KDR “Vascular endothelial growth factor receptor 2 inhibitor” CHEMBL3545155
Target PDGFRB “Platelet-derived growth factor receptor beta inhibitor” CHEMBL3545155