Drugs / Quabodepistat

Trials 7 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 12 trials
Phase 1 NCT07314320 Nov → Dec 2023 Otsuka Pharmaceutical Development & Commercialization, Inc. Completed No outcome recorded
Phase 1 NCT07542847 Sep → Nov 2022 Otsuka Pharmaceutical Development & Commercialization, Inc. Completed No outcome recorded
Phase 1/21 trial
Phase 1/2 NCT03678688 Oct 2018 → Feb 2022 pulmonary tuberculosis Otsuka Pharmaceutical Development & Commercialization, Inc. Completed No outcome recorded
Phase 23 trials
Phase 2 NCT06114628 Jan 2024 → Feb 2027 expected pulmonary tuberculosis University College, London Recruiting No outcome recorded
Phase 2 NCT05971602 Jul 2023 → Feb 2025 pulmonary tuberculosis Gates Medical Research Institute Terminated No outcome recorded
Phase 2 NCT05221502 Apr 2022 → Apr 2024 pulmonary tuberculosis Otsuka Pharmaceutical Development & Commercialization, Inc. Completed No outcome recorded
Phase 31 trial
Phase 3 NCT07209761 Oct 2025 → May 2027 expected pulmonary tuberculosis Otsuka Pharmaceutical Development & Commercialization, Inc. Recruiting No outcome recorded

Press releases naming this drug 6 releases

DateIssuerRelease
2025-11-06 Otsuka Pharmaceutical Development & Commercialization, Inc. Otsuka Announces First Participants Enrolled in Phase 3 Clinical Trial Evaluating Investigational Compound Quabodepistat for Drug-resistant Pulmonary Tuberculosis otsuka.co.jp
2025-11-06 Otsuka Pharmaceutical Development & Commercialization, Inc. Otsuka Announces First Participants Enrolled in Phase 3 Clinical Trial Evaluating Investigational Compound Quabodepistat for Drug-resistant Pulmonary Tuberculosis otsuka-us.com
2021-08-10 Otsuka Pharmaceutical Development & Commercialization, Inc. Otsuka Awarded Grant for Phase 2 Trial Combining Novel Anti-Tuberculosis Compound OPC-167832 with Delamanid and Bedaquiline otsuka.co.jp
2021-08-09 Otsuka Pharmaceutical Development & Commercialization, Inc. Otsuka Awarded Grant for Phase 2 Trial Combining Novel Anti-Tuberculosis Compound OPC-167832 with Delamanid and Bedaquiline otsuka-us.com
2018-01-29 Otsuka Pharmaceutical Development & Commercialization, Inc. Otsuka Awarded Grant to Advance Development of Novel Anti-Tuberculosis Compound OPC-167832 with Delamanid otsuka.co.jp
2018-01-29 Otsuka Pharmaceutical Development & Commercialization, Inc. Otsuka Awarded Grant to Advance Development of Novel Anti-Tuberculosis Compound OPC-167832 with Delamanid otsuka-us.com

Evidence & citations 6 cited values

Every value below carries the sentence it was read from. 9 sources stand behind the page.

FieldValueCited text
Known as Quabodepistat Quabodepistat in combination with delamanid and bedaquiline in participants with drug-susceptible pulmonary tuberculosis: protocol for a multicenter, phase 2b/c, open-label,...” PMID 38243296 Jan 2024
3

Quabodepistat (formerly OPC-167832) showed potent activity in preclinical studies and in the first stage of an early bactericidal activity study in adults with smear-positive,...” PMID 39612928 Nov 2024

“Bedaquiline 400 mg once daily for 2 weeks then 100 mg once daily for 15 weeks + Pretomanid 200 mg QD for 17 weeks + Quabodepistat 30 mg once daily for 17 weeks + Moxifloxacin...” NCT07209761

NCT06114628

Known as OPC-167832 “Quabodepistat (formerly OPC-167832) showed potent activity in preclinical studies and in the first stage of an early bactericidal activity study in adults with smear-positive,...” PMID 39612928 Nov 2024
3

NCT05971602

NCT07542847

NCT07314320

Known as QBS “Quabodepistat (QBS) is a newly discovered inhibitor of decaprenylphosphoryl-β-D-ribose-2'-oxidase, an essential enzyme for Mycobacterium tuberculosis to synthesize key...” PMID 38243296 Jan 2024
Action Inhibit inhibitor of decaprenylphosphoryl-β-D-ribose-2'-oxidase” PMID 38243296 Jan 2024
Modality Small molecule CHEMBL5095080
Route Oral “This trial will evaluate the safety, tolerability, pharmacokinetics (PK), and efficacy of multiple oral doses of OPC-167832 in participants with uncomplicated, smear-positive,...” NCT03678688