Drugs / Filibuvir
last change Jan 2012 re-read 2 minutes ago

Filibuvir

also known as PF-00868554 · PF-868554

Small molecule targets CYP3A4 via inhibition

Developed for
hepatitis C virus infection · chronic hepatitis C virus infection
Investigated by
Pfizer

Trials 10 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 18 trials
Phase 1 NCT01210404 Feb → May 2011 chronic hepatitis C virus infection Pfizer Completed No outcome recorded
Phase 1 NCT00918476 Jun 2010 → Feb 2011 hepatitis C virus infection Pfizer Completed No outcome recorded
Phase 1 NCT00861458 Apr → Jun 2009 hepatitis C virus infection Pfizer Completed No outcome recorded
Phase 1 NCT00875628 Apr 2009 Pfizer Terminated No outcome recorded
Phase 1 NCT00823745 Jan → Feb 2009 hepatitis C virus infection Pfizer Completed No outcome recorded
Phase 1 NCT00671671 Apr → Dec 2008 hepatitis C virus infection Pfizer Completed No outcome recorded
Phase 1 NCT00651027 Feb → Sep 2008 hepatitis C virus infection Pfizer Completed No outcome recorded
Phase 1 NCT00445315 Jan 2007 → Jun 2008 hepatitis C virus infection Pfizer Completed No outcome recorded
Phase 22 trials
Phase 2 NCT00987337 Nov 2009 → Jan 2012 hepatitis C virus infection Pfizer Completed No outcome recorded
Phase 2 NCT00720434 Aug 2008 → Mar 2010 chronic hepatitis C virus infection Pfizer Completed No outcome recorded
Also used as a comparator or background therapy in 1 trial
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1 NCT01051232 Comparator Feb → Apr 2010 Pfizer Completed No outcome recorded

Evidence & citations 7 cited values

Every value below carries the sentence it was read from. 11 sources stand behind the page.

FieldValueCited text
Known as Filibuvir “PF-00868554 (Filibuvir) following single oral administrations of PF-00868554 (Filibuvir) under fasting conditions in Japanese healthy adult volunteers” NCT01051232
4

“Antiviral activity of the hepatitis C virus polymerase inhibitor filibuvir in genotype 1-infected patients.” PMID 21488067 Jul 2011

NCT00987337

NCT00918476

NCT01210404

Known as PF-00868554 PF-00868554 (Filibuvir) following single oral administrations of PF-00868554 (Filibuvir) under fasting conditions in Japanese healthy adult volunteers” NCT01051232
5

“Single dose of 750 mg PF-00868554 as a solution and tablets.” NCT00861458

NCT00720434

NCT00875628

NCT00823745

NCT00445315

Known as PF-868554 ClinicalTrials.gov intervention name — accepted as the source's own label NCT00651027
Action Inhibit “non-nucleoside inhibitor filibuvir” PMID 21488067 Jul 2011
Modality Small molecule “non-nucleoside inhibitor filibuvir” PMID 21488067 Jul 2011
Route Oral “multiple oral doses of PF-00868554” NCT00445315
Target CYP3A4 “Filibuvir, a CYP3A4 inhibitor” NCT01210404