Drugs / Pecavaptan
last change Aug 2025 re-read 2 minutes ago

Pecavaptan

also known as BAY1753011

Small molecule targets AVPR1A, AVPR2 via inhibition

Developed for
heart failure
Investigated by
Bayer

Trials 2 · a red edge is where a trial was stopped

2020202120222023202420252026
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 11 trial
Phase 1 NCT05599997 Nov 2019 → Jan 2021 congestive heart failure, impaired renal function disease Bayer Completed No outcome recorded
Phase 21 trial
Phase 2 NCT03901729 May 2019 → Apr 2021 heart failure Bayer Completed No outcome recorded

Evidence & citations 7 cited values

Every value below carries the sentence it was read from. 5 sources stand behind the page.

FieldValueCited text
Known as pecavaptan “A multicentre, randomized, double-blind, active and placebo-controlled study of pecavaptan, a dual V1a/V2 vasopressin receptor antagonist, in patients with acute heart failure:...” PMID 40788619 Aug 2025
1

NCT05599997

Known as BAY1753011 “Pecavaptan (BAY1753011)” NCT05599997
Action Inhibit “pecavaptan, a novel, balanced dual-acting V1a/V2 vasopressin antagonist” PMID 33188886 Oct 2020
2

“Vasopressin V1a receptor antagonist” CHEMBL4594444

“Vasopressin V2 receptor antagonist” CHEMBL4594444

Modality Small molecule CHEMBL4594444
Route Oral “Tablet; 30mg or 5mg unit; 30mg once daily in the morning; OralNCT03901729
Target AVPR1A “Vasopressin V1a receptor antagonist” CHEMBL4594444
Target AVPR2 “Vasopressin V2 receptor antagonist” CHEMBL4594444