Drugs / ISIS 416858
last change Jul 2019 re-read 2 minutes ago

ISIS 416858

also known as FXI-ASO · IONIS-FXIRX · ISIS-FXIRx

Antisense oligonucleotide targets F11 via inhibition

Developed for
end stage renal failure · venous thromboembolism
Investigated by
Ionis Pharmaceuticals, Inc. · Bayer

Trials 3 · a red edge is where a trial was stopped

201320142015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 2 NCT03358030 Dec 2017 → Jul 2019 end stage renal failure Ionis Pharmaceuticals, Inc. Completed No outcome recorded
Phase 2 NCT02553889 Oct 2015 → Nov 2016 end stage renal failure Ionis Pharmaceuticals, Inc. Completed No outcome recorded
Phase 2 NCT01713361 Oct 2012 → May 2014 venous thromboembolism Ionis Pharmaceuticals, Inc. Completed No outcome recorded

Evidence & citations 8 cited values

Every value below carries the sentence it was read from. 4 sources stand behind the page.

FieldValueCited text
Known as ISIS 416858 “FXI-ASO (ISIS 416858) is a second-generation antisense oligonucleotide that specifically reduces factor XI levels.” PMID 25482425 Dec 2014
2

NCT03358030

NCT02553889

Known as FXI-ASO FXI-ASO (ISIS 416858) is a second-generation antisense oligonucleotide that specifically reduces factor XI levels.” PMID 25482425 Dec 2014
Known as IONIS-FXIRX “A Phase 2, Randomized, Double-Blind, Placebo-Controlled Study of the Safety, Pharmacokinetics, and Pharmacodynamics of Multiple Doses of ISIS 416858 (IONIS-FXIRX, an Antisense...” NCT03358030
Known as ISIS-FXIRx ClinicalTrials.gov intervention name — accepted as the source's own label NCT01713361
Action Inhibit “specifically reduces factor XI levels” PMID 25482425 Dec 2014
Modality Antisense oligonucleotide “FXI-ASO (ISIS 416858) is a second-generation antisense oligonucleotide that specifically reduces factor XI levels.” PMID 25482425 Dec 2014
Route Subcutaneous subcutaneously administered” NCT01713361
Target F11 “specifically reduces factor XI levels” PMID 25482425 Dec 2014