Drugs / Pexacerfont
last change Sep 2015 re-read 2 minutes ago

Pexacerfont

also known as BMS-562086 · CRF1 ANTAGONIST · Dpc-a69448

Small molecule targets CRHR1 via inhibition

Developed for
generalized anxiety disorder · irritable bowel syndrome · major depressive disorder · alcohol dependence · anxiety disorder
Investigated by
Bristol-Myers Squibb · National Institute on Drug Abuse (NIDA)

Trials 4 · a red edge is where a trial was stopped

2006200720082009201020112012201320142015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 01 trial
Phase 0 NCT01656577 Jun 2012 → Sep 2015 National Institute on Drug Abuse (NIDA) Terminated No outcome recorded
Phase 1/21 trial
Phase 1/2 NCT00135421 Nov 2005 → Oct 2007 major depressive disorder Bristol-Myers Squibb Completed No outcome recorded
Phase 21 trial
Phase 2 NCT00399438 Dec 2006 → Oct 2007 irritable bowel syndrome Bristol-Myers Squibb Completed No outcome recorded
Phase 2/31 trial
Phase 2/3 NCT00481325 Jul 2007 → Mar 2008 generalized anxiety disorder Bristol-Myers Squibb Completed No outcome recorded
Also used as a comparator or background therapy in 1 trial
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 2 NCT01227980 Comparator Oct 2010 → Jul 2014 alcohol dependence, anxiety disorder National Institute on Alcohol Abuse and Alcoholism (NIAAA) Completed No outcome recorded

Evidence & citations 8 cited values

Every value below carries the sentence it was read from. 7 sources stand behind the page.

FieldValueCited text
Known as Pexacerfont ClinicalTrials.gov intervention name — accepted as the source's own label NCT00135421
3

NCT01656577

NCT01227980

NCT00481325

Known as BMS-562086 ClinicalTrials.gov intervention name — accepted as the source's own label NCT00399438
Known as CRF1 ANTAGONIST ChEMBL registry synonym — accepted as the source's own label CHEMBL482950
Known as Dpc-a69448 ChEMBL registry synonym — accepted as the source's own label CHEMBL482950
Action Inhibit “Corticotropin releasing factor receptor 1 antagonist” CHEMBL482950
1

“pexacerfont, a selective CRF-1 receptor antagonist” PMID 20455246 May 2010

Modality Small molecule CHEMBL482950
Route Oral OralNCT00135421
Target CRHR1 “Corticotropin releasing factor receptor 1 antagonist” CHEMBL482950