Drugs / DELANZOMIB
last change Jan 2017 re-read 2 minutes ago

DELANZOMIB

also known as CEP 18770 · CIP 18770 · CT 47098 · NPH 007098

Small molecule

Developed for
plasma cell myeloma · cancer · non-Hodgkin lymphoma
Investigated by
Cephalon · Ethical Oncology Science · Teva Branded Pharmaceutical Products R&D, Inc.

Trials 3 · a red edge is where a trial was stopped

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PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 11 trial
Phase 1 NCT00572637 Nov 2007 → Mar 2010 cancer, non-Hodgkin lymphoma Ethical Oncology Science Completed No outcome recorded
Phase 1/22 trials
Phase 1/2 NCT01348919 Aug 2011 → Mar 2013 plasma cell myeloma Teva Branded Pharmaceutical Products R&D, Inc. Completed No outcome recorded
Phase 1/2 NCT01023880 Jan 2010 → Nov 2012 plasma cell myeloma Cephalon Terminated No outcome recorded

Evidence & citations 8 cited values

Every value below carries the sentence it was read from. 5 sources stand behind the page.

FieldValueCited text
Known as DELANZOMIB ChEMBL registry synonym — accepted as the source's own label CHEMBL270515
Known as CEP 18770 “This is an open-label, multicenter, dose-escalating study to determine the MTD and dose limiting toxicities (DLTs) of CEP 18770, a novel proteasome inhibitor.” NCT00572637
3

NCT01348919

NCT00572637

NCT01023880

Known as CIP 18770 ChEMBL registry synonym — accepted as the source's own label CHEMBL270515
Known as CT 47098 ChEMBL registry synonym — accepted as the source's own label CHEMBL270515
Known as NPH 007098 ChEMBL registry synonym — accepted as the source's own label CHEMBL270515
Action Inhibit “CEP 18770, a novel proteasome inhibitor” NCT00572637
Modality Small molecule “Delanzomib (CEP-18770), a reversible P2 threonine boronic acid proteasome (β5/β1 subunits) inhibitor” PMID 28140719 Jan 2017
Route Intravenous “Patients will be treated intravenously with CEP 18770 on days 1, 4, 8, and 11 of a 21-day cycle period.” NCT00572637