Drugs / IZORLISIB
last change Apr 2026 re-read 2 minutes ago

IZORLISIB

also known as MEN1611 · CH5132799 · CH5132799-000 · PA-799

Small molecule targets PIK3CA via inhibition

Developed for
breast cancer · cancer · colorectal cancer
Investigated by
Menarini Group · Chugai Pharma Europe Ltd. · MedSIR

Trials 4 · a red edge is where a trial was stopped

20112012201320142015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 12 trials
Phase 1 NCT03767335 Nov 2018 → Feb 2024 breast cancer Menarini Group Completed No outcome recorded
Phase 1 NCT01222546 Aug 2010 → Nov 2012 cancer Chugai Pharma Europe Ltd. Completed No outcome recorded
Phase 1/21 trial
Phase 1/2 NCT04495621 Jul 2020 → Jan 2024 colorectal cancer Menarini Group Completed No outcome recorded
Phase 21 trial
Phase 2 NCT05810870 May 2023 → Apr 2026 overdue breast cancer MedSIR Active not recruiting No outcome recorded

Evidence & citations 9 cited values

Every value below carries the sentence it was read from. 5 sources stand behind the page.

FieldValueCited text
Known as IZORLISIB ChEMBL registry synonym — accepted as the source's own label CHEMBL1684984
Known as CH5132799 ClinicalTrials.gov intervention name — accepted as the source's own label NCT01222546
Known as CH5132799-000 ChEMBL registry synonym — accepted as the source's own label CHEMBL1684984
Known as MEN1611 ClinicalTrials.gov intervention name — accepted as the source's own label NCT03767335
2

NCT05810870

NCT04495621

Known as PA-799 ChEMBL registry synonym — accepted as the source's own label CHEMBL1684984
Action Inhibit “MEN1611 is an investigational drug which blocks a protein called PI3K” NCT03767335
Modality Small molecule CHEMBL1684984
Route Oral “administered orally” NCT01222546
Target PIK3CA “PI3K alpha inhibitor MEN1611 selectively binds to and inhibits PIK3CA and its mutated forms in the PI3K/Akt (protein kinase B)/mammalian target of rapamycin (mTOR) pathway.” NCT05810870