Drugs / Duligotuzumab
last change Apr 2018 re-read 2 minutes ago

Duligotuzumab

also known as MEHD7945A · Duligotumab · RG-7597

Monoclonal antibody targets EGFR, ERBB3 via inhibition

Developed for
head and neck cancer · colorectal cancer · epithelial neoplasm · neoplasm
Investigated by
Genentech, Inc.

Trials 5 · a red edge is where a trial was stopped

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PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 13 trials
Phase 1 NCT01986166 Nov 2013 → Jan 2016 neoplasm Genentech, Inc. Completed No outcome recorded
Phase 1 NCT01911598 Sep 2013 → Jun 2017 head and neck cancer Genentech, Inc. Completed No outcome recorded
Phase 1 NCT01207323 Nov 2010 → Dec 2013 epithelial neoplasm Genentech, Inc. Completed No outcome recorded
Phase 22 trials
Phase 2 NCT01652482 Oct 2012 → Nov 2014 colorectal cancer Genentech, Inc. Completed No outcome recorded
Phase 2 NCT01577173 Jul 2012 → Jun 2015 head and neck cancer Genentech, Inc. Completed No outcome recorded

Evidence & citations 9 cited values

Every value below carries the sentence it was read from. 7 sources stand behind the page.

FieldValueCited text
Known as Duligotuzumab “Phase II Study of the Dual EGFR/HER3 Inhibitor Duligotuzumab (MEHD7945A) versus Cetuximab in Combination with FOLFIRI in Second-Line RAS Wild-Type Metastatic Colorectal Cancer.” PMID 29506988 Mar 2018
Known as Duligotumab ChEMBL registry synonym — accepted as the source's own label CHEMBL3137345
Known as MEHD7945A ClinicalTrials.gov intervention name — accepted as the source's own label NCT01652482
4

NCT01207323

NCT01577173

NCT01986166

NCT01911598

Known as RG-7597 ChEMBL registry synonym — accepted as the source's own label CHEMBL3137345
Action Inhibit “Phase II Study of the Dual EGFR/HER3 Inhibitor Duligotuzumab (MEHD7945A)” PMID 29506988 Mar 2018
1

“Receptor tyrosine-protein kinase erbB-3 inhibitor” CHEMBL3137345

Modality Monoclonal antibody CHEMBL3137345
Route Intravenous “Participants will receive intravenous (IV) infusion of MEHD7945A in escalating doses Q2W” NCT01207323
Target EGFR “Duligotuzumab is a dual-action antibody directed against EGFR and HER3.” PMID 29506988 Mar 2018
Target ERBB3 “Receptor tyrosine-protein kinase erbB-3 inhibitor” CHEMBL3137345