Drugs / saracatinib
last change Jun 2025 re-read 2 minutes ago

saracatinib

Small molecule targets ABL1, ACVR1, FYN, SRC via inhibition

Developed for
alcohol-related disorders · Alzheimer disease · breast cancer · hormone-resistant prostate carcinoma · lung lymphangioleiomyomatosis · neoplasm · non-small cell lung carcinoma · adult fibrosarcoma
+39 more · adult liposarcoma · bone neoplasm · cancer · colon adenocarcinoma · combined thymoma · dermatofibrosarcoma protuberans · estrogen-receptor negative breast cancer · fibrodysplasia ossificans progressiva · gastric adenocarcinoma · gastroesophageal junction adenocarcinoma · hypopharynx squamous cell carcinoma · larynx verrucous carcinoma · leiomyosarcoma · male breast carcinoma · malignant epithelial tumor of ovary · malignant pancreatic neoplasm · melanoma · metastatic squamous cell carcinoma · nasal cavity and paranasal sinus squamous cell carcinoma · nasopharyngeal squamous cell carcinoma · oropharynx squamous cell carcinoma · ovarian cancer · pancreatic adenocarcinoma · Parkinson disease · pleural neoplasm · progesterone-receptor negative breast cancer · prostate cancer · rectum adenocarcinoma · rhabdomyosarcoma · small cell lung carcinoma · tongue cancer · undifferentiated pleomorphic sarcoma · uterine carcinosarcoma · uterine corpus endometrial stromal sarcoma · verrucous carcinoma of oral cavity · fallopian tube cancer · idiopathic pulmonary fibrosis · osteosarcoma · primary peritoneal carcinoma
Investigated by
National Cancer Institute (NCI) · AstraZeneca · Yale University · Brigham and Women's Hospital · National Institute on Alcohol Abuse and Alcoholism (NIAAA) · Stanford University
+19 more · University of Cincinnati · Alzheimer's Therapeutic Research Institute · Amsterdam UMC, location VUmc · Baylor College of Medicine · Innovative Medicines Initiative · Joyce Marie Slingerland, MD · King's College Hospital NHS Trust · King's College London · Klinikum Garmisch-Patenkirchen · Loyola University · NCIC Clinical Trials Group · National Institute of Neurological Disorders and Stroke (NINDS) · National Institutes of Health (NIH) · Royal National Orthopaedic Hospital NHS Trust · Stephen M. Strittmatter · Tony Eissa · University of Oxford · University of South Florida · University of Texas

Trials 31 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 01 trial
Phase 0 NCT03661125 Apr 2019 → Sep 2021 Parkinson disease King's College London Unknown No outcome recorded
Phase 110 trials
Phase 1 NCT02732587 Nov 2015 → Mar 2016 alcohol-related disorders Yale University Completed No outcome recorded
Phase 1 NCT02262026 Nov 2014 → Apr 2019 alcohol dependence Yale University Completed No outcome recorded
Phase 1 NCT02116712 Aug 2014 → Jun 2015 lung lymphangioleiomyomatosis Tony Eissa Completed No outcome recorded
Phase 1 NCT01864655 Jul 2013 → Mar 2014 Alzheimer disease Stephen M. Strittmatter Completed No outcome recorded
Phase 1 NCT01000896 Jan → Sep 2010 malignant epithelial tumor of ovary, non-small cell lung carcinoma AstraZeneca Withdrawn No outcome recorded
Phase 1 NCT00853983 Mar → Apr 2009 AstraZeneca Completed No outcome recorded
Phase 1 NCT00771979 Nov 2008 → Mar 2009 AstraZeneca Completed No outcome recorded
Phase 1 NCT00704366 Jun 2008 → Jan 2011 cancer AstraZeneca Completed No outcome recorded
Phase 1 NCT00475956 May 2007 → Oct 2008 neoplasm AstraZeneca Completed No outcome recorded
Phase 1 NCT00496028 Mar 2007 → Jan 2010 neoplasm AstraZeneca Completed No outcome recorded
Phase 1/22 trials
Phase 1/2 NCT01216176 Oct 2008 → Feb 2018 breast cancer Joyce Marie Slingerland, MD Completed No outcome recorded
Phase 1/2 NCT00265876 Apr 2006 → Jan 2009 malignant pancreatic neoplasm NCIC Clinical Trials Group Completed No outcome recorded
Phase 218 trials
Phase 2 NCT04307953 Aug 2020 → May 2025 fibrodysplasia ossificans progressiva Amsterdam UMC, location VUmc Unknown No outcome recorded
Phase 2 NCT02955186 May 2017 → Apr 2019 alcohol-related disorders Yale University Completed No outcome recorded
Phase 2 NCT02737202 Apr 2016 → Jul 2019 lung lymphangioleiomyomatosis Baylor College of Medicine Terminated No outcome recorded
Phase 2 NCT02167256 Dec 2014 → Feb 2018 Alzheimer disease Yale University Completed No outcome recorded
Phase 2 NCT01267266 Dec 2010 → Sep 2012 hormone-resistant prostate carcinoma National Cancer Institute (NCI) Terminated No outcome recorded
Phase 2 NCT00735917 Oct 2008 → Apr 2011 pancreatic adenocarcinoma National Cancer Institute (NCI) Completed No outcome recorded
Phase 2 NCT00718809 Jun 2008 → Aug 2010 combined thymoma National Cancer Institute (NCI) Terminated No outcome recorded
Phase 2 NCT00610714 Apr 2008 → Aug 2009 ovarian cancer AstraZeneca Completed No outcome recorded
Phase 2 NCT00659360 Feb 2008 → Jan 2009 adult fibrosarcoma, adult liposarcoma, dermatofibrosarcoma protuberans, leiomyosarcoma +4 National Cancer Institute (NCI) Completed No outcome recorded
Phase 2 NCT00638937 Feb 2008 → Jun 2013 non-small cell lung carcinoma National Cancer Institute (NCI) Completed No outcome recorded
Also used as a comparator or background therapy in 4 trials
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1/21 trial
Phase 1/2 NCT04598919 Comparator Nov 2020 → Sep 2024 overdue idiopathic pulmonary fibrosis National Jewish Health Active not recruiting No outcome recorded
Phase 22 trials
Phase 2 NCT02085603 Comparator Mar 2014 → Jan 2018 cancer Sheffield Teaching Hospitals NHS Foundation Trust Completed No outcome recorded
Phase 2 NCT00752206 Comparator Mar 2009 → Aug 2017 osteosarcoma Sarcoma Alliance for Research through Collaboration Terminated No outcome recorded
Phase 2/31 trial
Phase 2/3 NCT01196741 Comparator Mar 2011 → Nov 2012 fallopian tube cancer, ovarian cancer, primary peritoneal carcinoma University College, London Completed No outcome recorded

Evidence & citations 9 cited values

Every value below carries the sentence it was read from. 38 sources stand behind the page.

FieldValueCited text
Known as saracatinib “The study includes the use of saracatinib, an investigational drug originally developed to treat certain types of cancers, in the treatment of IPF in a Phase 1b/2a clinical trial.” NCT04598919
24

Saracatinib (AZD0530) is a selective, oral Src inhibitor that has demonstrated antitumour activity in preclinical studies.” PMID 22415795 Mar 2012

“Src inhibitor saracatinib (AZD0530)” PMID 21170669 Dec 2010

“AZD0530 (also called saracatinib)” NCT01216176

NCT02737202

NCT00669019

NCT00659360

NCT02085603

NCT01196741

NCT00397878

NCT00513071

NCT00528645

NCT02955186

NCT03661125

NCT01267266

NCT00735917

NCT00559507

NCT00638937

NCT02116712

NCT00718809

NCT00607594

NCT00752206

NCT02732587

NCT01864655

NCT00513435

Known as AZ-10353926 ChEMBL registry synonym — accepted as the source's own label CHEMBL217092
Known as AZD0530 “The purpose of this study is to investigate whether the addition of the Src inhibitor saracatinib (AZD0530) to weekly paclitaxel improves efficacy” NCT01196741
19

AZD0530 (Saracatinib) 50 mg Tablet Pink Round 7.0 mm ADM P/5406/49. Two tablets to be taken every morning for 14 days.” NCT03661125

“A Placebo-Controlled Study of Saracatinib (AZD0530) in Patients With Recurrent Osteosarcoma Localized to the Lung” NCT00752206

“To estimate the disease control rate of AZD0530 (saracatinib) in patients with metastatic breast cancer.” NCT00559507

“patients with AZD0530 (saracatinib) in patients with advanced non-small cell lung cancer” NCT00638937

“saracatinib/AZD0530 (placebo or 125 mg/day)” NCT02955186

AZD0530NCT00659360

NCT00771979

NCT02167256

NCT00558272

NCT01000896

NCT02262026

NCT00610714

NCT00704366

NCT00265876

NCT01216176

NCT00475956

NCT04307953

NCT00496028

NCT00853983

Known as Saracatinib fumarate ChEMBL registry synonym — accepted as the source's own label CHEMBL217092
Action Inhibit “Tyrosine-protein kinase ABL inhibitor” CHEMBL217092
1

“Src inhibitor” PMID 21170669 Dec 2010

Modality Small molecule CHEMBL217092
Route Oral “Patients receive oral AZD0530 once daily on days 1-28” NCT00265876
Target ABL1 “Tyrosine-protein kinase ABL inhibitor” CHEMBL217092
Target SRC Src inhibitor” PMID 21170669 Dec 2010