Drugs / fevipiprant
last change Dec 2021 re-read 2 minutes ago

fevipiprant

also known as QAW039 · NVP-QAW039

Small molecule targets PTGDR2 via inhibition

Developed for
asthma · allergic rhinitis · atopic eczema · chronic asthma · chronic obstructive pulmonary disease · nasal cavity polyp
Investigated by
Novartis Pharmaceuticals

Trials 16 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 12 trials
Phase 1 NCT03087942 Jul 2017 → Aug 2018 impaired renal function disease Novartis Pharmaceuticals Completed No outcome recorded
Phase 1 NCT03048448 May 2017 → Apr 2019 Novartis Pharmaceuticals Completed No outcome recorded
Phase 29 trials
Phase 2 NCT03989635 Oct 2019 → Jun 2021 asthma, eosinophil disorder Novartis Pharmaceuticals Withdrawn No outcome recorded
Phase 2 NCT03810183 May 2019 → Jan 2020 chronic obstructive pulmonary disease Novartis Pharmaceuticals Terminated No outcome recorded
Phase 2 NCT03650400 May → Dec 2019 asthma Novartis Pharmaceuticals Terminated No outcome recorded
Phase 2 NCT01785602 Jun 2013 → Nov 2014 atopic eczema Novartis Pharmaceuticals Completed No outcome recorded
Phase 2 NCT01836471 May 2013 → Feb 2016 asthma Novartis Pharmaceuticals Completed No outcome recorded
Phase 2 NCT01804400 Oct 2012 → Oct 2013 allergic rhinitis Novartis Pharmaceuticals Completed No outcome recorded
Phase 2 NCT01545726 Feb 2012 → Jun 2013 asthma Novartis Pharmaceuticals Completed No outcome recorded
Phase 2 NCT01437735 Aug 2011 → Nov 2013 asthma Novartis Pharmaceuticals Completed No outcome recorded
Phase 2 NCT01253603 Nov 2010 → Sep 2011 chronic asthma Novartis Pharmaceuticals Completed No outcome recorded
Phase 35 trials
Phase 3 NCT03681093 Mar 2019 → May 2020 nasal cavity polyp Novartis Pharmaceuticals Completed No outcome recorded
Phase 3 NCT03629249 Dec 2018 → Feb 2020 asthma Novartis Pharmaceuticals Terminated No outcome recorded
Phase 3 NCT03052517 Mar 2017 → Feb 2020 asthma Novartis Pharmaceuticals Terminated No outcome recorded
Phase 3 NCT02555683 Dec 2015 → Oct 2019 asthma Novartis Pharmaceuticals Completed No outcome recorded
Phase 3 NCT02563067 Dec 2015 → Jul 2019 asthma Novartis Pharmaceuticals Completed No outcome recorded
Also used as a comparator or background therapy in 2 trials
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 3 NCT03215758 Comparator Nov 2017 → Jul 2019 asthma Novartis Pharmaceuticals Completed No outcome recorded
Phase 3 NCT03226392 Comparator Oct 2017 → Jul 2019 asthma Novartis Pharmaceuticals Completed No outcome recorded

Evidence & citations 7 cited values

Every value below carries the sentence it was read from. 24 sources stand behind the page.

FieldValueCited text
Known as fevipiprant “Dose-related efficacy and safety of fevipiprant (QAW039), an oral DP2 (CRTh2) receptor antagonist, was assessed in patients with allergic asthma uncontrolled by low-dose...” PMID 28838980 Aug 2017
9

Fevipiprant, an oral antagonist of the prostaglandin D2 receptor 2, reduced sputum eosinophils and improved lung function in phase 2 trials of patients with asthma.” PMID 32979986 Sep 2020

Fevipiprant is an oral, non-steroidal, highly selective, reversible antagonist of the DP2 receptor that inhibits the binding of PGD2 and its metabolites.” PMID 34895218 Dec 2021

“QAW039 (fevipiprant) 450 mg once daily for 6 weeks administered orally as a tablet + Standard of Care” NCT03810183

fevipiprant (QAW039), an antagonist of prostaglandin D2 receptor 2” PMID 27503237 Aug 2016

“The oral CRTh2 antagonist QAW039 (fevipiprant)” PMID 27354118 Jun 2016

fevipiprant (QAW039)” NCT03989635

NCT03048448

NCT03681093

NCT03650400

Known as NVP-QAW039 ChEMBL registry synonym — accepted as the source's own label CHEMBL3137332
Known as QAW039 “The overall purpose of this study was to provide long- term safety data for fevipiprant (QAW039) (Dose 1 and Dose 2), compared with placebo, when added to the Global Initiative...” NCT03052517
15

QAW039 (fevipiprant) 450 mg once daily for 6 weeks administered orally as a tablet + Standard of Care” NCT03810183

“Fevipiprant (QAW039) 150 mg once daily administered orally as tablet” NCT03681093

NCT03989635

NCT03629249

NCT01545726

NCT02563067

NCT01253603

NCT02555683

NCT03215758

NCT01785602

NCT01437735

NCT03226392

NCT01804400

NCT03087942

NCT01836471

Action Inhibit “QAW039, an oral chemoattractant receptor-homologous molecule expressed on Th2 cells (CRTh2) receptor antagonist” PMID 27354118 Jun 2016
1

“G protein-coupled receptor 44 antagonist” CHEMBL3137332

Modality Small molecule CHEMBL3137332
Route Oral “QAW039, an oral chemoattractant receptor-homologous molecule” PMID 27354118 Jun 2016
Target PTGDR2 “G protein-coupled receptor 44 antagonist” CHEMBL3137332