Drugs / MUBRITINIB
last change Sep 2003 re-read 3 minutes ago

MUBRITINIB

also known as TAK-165

Small molecule targets ERBB2 via inhibition

Developed for
breast neoplasm · kidney neoplasm · lung neoplasm · ovarian neoplasm · pancreatic neoplasm
Investigated by
Takeda

Trials 1

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PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1 NCT00034281 Jun 2002 → Sep 2003 breast neoplasm, kidney neoplasm, lung neoplasm, ovarian neoplasm +1 Takeda Completed No outcome recorded

Evidence & citations 5 cited values

Every value below carries the sentence it was read from. 2 sources stand behind the page.

FieldValueCited text
Known as MUBRITINIB ChEMBL registry synonym — accepted as the source's own label CHEMBL1614707 ↗
Known as TAK-165 ClinicalTrials.gov intervention name — accepted as the source's own label NCT00034281 ↗
Action Inhibit “TAK-165 is an active and selective inhibitor of tyrosine kinase activity of HER2” NCT00034281 ↗
1

“Receptor protein-tyrosine kinase erbB-2 inhibitor” CHEMBL1614707 ↗

Modality Small molecule — CHEMBL1614707 ↗
Target ERBB2 “Receptor protein-tyrosine kinase erbB-2 inhibitor” CHEMBL1614707 ↗