Drugs / Liafensine
last change Dec 2025 re-read 2 minutes ago

Liafensine

also known as BMS-820836 · Liafensina

Small molecule

Developed for
depressive disorder · major depressive disorder
Investigated by
Bristol-Myers Squibb · Denovo Biopharma LLC

Trials 6 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 12 trials
Phase 1 NCT01396252 Sep 2011 → May 2012 depressive disorder Bristol-Myers Squibb Completed No outcome recorded
Phase 1 NCT00892840 May 2009 → Nov 2010 depressive disorder Bristol-Myers Squibb Completed No outcome recorded
Phase 24 trials
Phase 2 NCT05113771 Jun 2022 → Feb 2024 Denovo Biopharma LLC Completed No outcome recorded
Phase 2 NCT01361555 Aug 2011 → Oct 2013 major depressive disorder Bristol-Myers Squibb Terminated No outcome recorded
Phase 2 NCT01369095 Jul 2011 → May 2013 depressive disorder Bristol-Myers Squibb Completed No outcome recorded
Phase 2 NCT01309945 Apr 2011 → Jan 2013 depressive disorder Bristol-Myers Squibb Completed No outcome recorded
Also used as a comparator or background therapy in 1 trial
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1 NCT00964912 Comparator Jul 2008 → Apr 2009 depressive disorder Bristol-Myers Squibb Completed No outcome recorded

Evidence & citations 6 cited values

Every value below carries the sentence it was read from. 9 sources stand behind the page.

FieldValueCited text
Known as Liafensine ClinicalTrials.gov intervention name — accepted as the source's own label NCT05113771
Known as BMS-820836 ClinicalTrials.gov intervention name — accepted as the source's own label NCT01361555
5

NCT00964912

NCT01309945

NCT01369095

NCT01396252

NCT00892840

Known as Liafensina ChEMBL registry synonym — accepted as the source's own label CHEMBL2364614
Action Inhibit “Liafensine, a triple reuptake inhibitor, may become a new precision medicine for treatment-resistant depression (TRD), a major unmet medical need.” PMID 40928787 Dec 2025
Modality Small molecule CHEMBL2364614
Route Oral Oral Solution, Oral” NCT00892840