Drugs / Clesacostat
last change Jul 2024 re-read 2 minutes ago

Clesacostat

also known as PF-05221304 · PF'1304

Small molecule

Developed for
NAFLD1 · metabolic dysfunction-associated steatohepatitis
Investigated by
Pfizer

Trials 9 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 16 trials
Phase 1 NCT03871439 Mar → May 2019 Pfizer Completed No outcome recorded
Phase 1 NCT03597217 Aug → Nov 2018 Pfizer Completed No outcome recorded
Phase 1 NCT03534648 Apr → Jul 2018 Pfizer Completed No outcome recorded
Phase 1 NCT03448172 Apr → May 2018 Pfizer Completed No outcome recorded
Phase 1 NCT03309202 Dec 2017 → Jun 2018 liver disease, severe congenital Pfizer Completed No outcome recorded
Phase 1 NCT02871037 Aug 2016 → Mar 2017 Pfizer Completed No outcome recorded
Phase 23 trials
Phase 2 NCT04399538 Aug 2020 → Mar 2022 NAFLD1, metabolic dysfunction-associated steatohepatitis Pfizer Completed No outcome recorded
Phase 2 NCT04321031 Jun 2020 → Jan 2024 NAFLD1, metabolic dysfunction-associated steatohepatitis Pfizer Completed No outcome recorded
Phase 2 NCT03776175 Jan → Sep 2019 NAFLD1 Pfizer Completed No outcome recorded
Also used as a comparator or background therapy in 2 trials
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 11 trial
Phase 1 NCT04395950 Comparator Dec 2020 → Aug 2021 NAFLD1, metabolic dysfunction-associated steatohepatitis Columbia University Withdrawn No outcome recorded
Phase 21 trial
Phase 2 NCT03248882 Comparator Aug 2017 → Feb 2019 NAFLD1, metabolic dysfunction-associated steatohepatitis Pfizer Completed No outcome recorded

Press releases naming this drug 1 release

DateIssuerRelease
2022-05-26 Pfizer Pfizer Granted FDA Fast Track Designation for Ervogastat/Clesacostat Combination for the Treatment of Non-Alcoholic Steatohepatitis (NASH) pfizer.com

Evidence & citations 6 cited values

Every value below carries the sentence it was read from. 13 sources stand behind the page.

FieldValueCited text
Known as clesacostat “with Clesacostat (PF-05221304), an acetyl coA carboxylase inhibitor (ACCi) in patients with NAFLD/NASH.” PMID 39048608 Jul 2024
1

“acetyl-coenzyme A carboxylase inhibitor (ACCi, PF-05221304, clesacostat)” PMID 35354614 Mar 2022

Known as PF'1304 “The purpose of this study is to assess the effects of an investigational drug, PF-05221304 (PF'1304) on the way the liver handles fat.” NCT04395950
Known as PF-05221304 ClinicalTrials.gov intervention name — accepted as the source's own label NCT03871439
10

NCT04395950

NCT04321031

NCT03776175

NCT04399538

NCT03597217

NCT03448172

NCT03309202

NCT02871037

NCT03534648

NCT03248882

Action Inhibit “Clesacostat (PF-05221304), an acetyl coA carboxylase inhibitor (ACCi)” PMID 39048608 Jul 2024
Modality Small molecule Small molecule inhibitors of the terminal step in intrahepatic triglyceride synthesis (diacylglycerol acyltransferase 2 inhibitor (DGAT2i, PF-06865571, ervogastat)) and...” PMID 35354614 Mar 2022
Route Oral Oral Doses” NCT02871037