drugset / Trial / NCT01249118

An Absolute Bioavailability Study in Healthy Participants Comparing Oral to Intravenous Administration of GDC-0973 (Cobimetinib)

NCT01249118

Phase 1 Completed 13 enrolled Genentech, Inc.
RandomizedCrossoverOpen-labelBasic science

Summary

The primary objective of Part 1 of this study is to evaluate the safety and tolerability of the intravenous (IV) dose of GDC-0973. The primary objectives of Part 2 of this study are to evaluate the absolute bioavailability of GDC-0973 and to evaluate the pharmacokinetic (PK) of GDC-0973 following IV and oral administration. The secondary objective of Part 2 of this study is to evaluate the safety of GDC-0973 administered orally and intravenously.

Timeline

Start
2010-11
Primary completion
2011-01
Completion
2011-01

Drugs

EvaluationDrugModalityDoseRoute
Subject Cobimetinib Small molecule 2 mg Intravenous
Subject Cobimetinib Small molecule 20 mg Intravenous

Indications

No indication recorded.